SCHEMBL29119

SCHEMBL29119

COc1ccc2c(ccn2[Si](C(C)C)(C(C)C)C(C)C)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.54
ROCK1 Q13464 1/20 0.45
POLB P06746 1/20 0.43
HTR6 P50406 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
SLC6A2 P23975 2/20 0.41
TUBB1 Q9H4B7 1/20 0.41
PDGFRB P09619 1/20 0.40
PDGFRA P16234 1/20 0.40
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
PTGS2 P35354 3/20 0.40
PTGS1 P23219 2/20 0.40
AKR1C3 P42330 2/20 0.40
AKR1C2 P52895 2/20 0.40
CYP1A2 P05177 2/20 0.40
TSHR P16473 2/20 0.40
CDC42 P60953 1/20 0.40
RAC1 P63000 1/20 0.40
SLC22A6 Q4U2R8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28979 0.78 HTR2A (0.49) HTR2CROCK1SLC6A2CYP1A2CYP2A6
SCHEMBL2502244 0.77 KDM4E (0.36) HTR2CCYP1A2MAPT
SCHEMBL30967900 0.77 HTR2A (0.50) HTR2CROCK1HTR6SLC6A2CYP2A6
SCHEMBL2073701 0.77 PRKCI (0.53) HTR2CPOLBMAPTLMNA
SCHEMBL850727 0.77 HTR2C (0.50) HTR2CSLC6A2SLC6A4PRMT5MAPT
SCHEMBL3327014 0.77 MAPT (0.33) HTR2CMAPT
SCHEMBL30949143 0.77 HTR2A (0.50) HTR2CSLC6A2SLC6A4PRMT5MAPT
SCHEMBL29533363 0.75 HTR2C (0.35) HTR2CROCK1CYP1A2MAPTCYP2C9
SCHEMBL1856356 0.75 KDM4E (0.46) POLBTUBB1MAPTLMNACYP2C9
SCHEMBL597518 0.75 HTR2C (0.58) HTR2CROCK1POLBHTR6L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012025760-A1 PROCESS FOR THE BORYLATION OF ARENES AND HETEROARYLS THE UNIVERSITY OF MANCHESTER (GB) 2012-03-01 WO disclosed