SCHEMBL2912265

SCHEMBL2912265

CCOC(=O)c1cnc2cc(N3CCN(CC)CC3)c(OC)cc2c1Nc1cc(C)ccc1F

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 8/20 0.58
KCNH2 Q12809 4/20 0.54
SCN5A Q14524 4/20 0.54
GAA P10253 2/20 0.49
MAPT P10636 2/20 0.49
THRB P10828 1/20 0.49
MEN1 O00255 1/20 0.47
LMNA P02545 1/20 0.47
MC4R P32245 1/20 0.47
HTT P42858 1/20 0.47
KMT2A Q03164 1/20 0.47
PTK2B Q14289 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2912359 0.93 CSF1R (0.63) CSF1RKCNH2SCN5AGAAMAPT
SCHEMBL2912181 0.91 KCNH2 (0.65) CSF1RKCNH2SCN5AGAAMAPT
SCHEMBL2911180 0.91 CSF1R (0.71) CSF1RKCNH2SCN5A
SCHEMBL2904655 0.90 CSF1R (0.59) CSF1RKCNH2SCN5AGAAMAPT
SCHEMBL2907777 0.90 KCNH2 (0.67) CSF1RKCNH2SCN5AGAAMEN1
SCHEMBL2907821 0.86 CSF1R (0.58) CSF1RKCNH2SCN5AGAAMAPT
SCHEMBL2910399 0.86 CSF1R (0.69) CSF1RKCNH2SCN5A
SCHEMBL2908740 0.86 KCNH2 (0.64) CSF1RKCNH2SCN5A
SCHEMBL2911044 0.85 CSF1R (0.69) CSF1RKCNH2SCN5AGAAMEN1
SCHEMBL2912778 0.85 KCNH2 (0.74) CSF1RKCNH2SCN5AGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed