SCHEMBL2913331

SCHEMBL2913331

Nc1nc(NCCCn2cc(C(=O)NC3CC3)c(-c3ccc(-n4ccnc4)cc3)c2)ccc1[N+](=O)[O-]

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.41
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
CD38 P28907 11/20 0.39
AXL P30530 1/20 0.35
FLT3 P36888 1/20 0.35
TYRO3 Q06418 1/20 0.35
MERTK Q12866 1/20 0.35
GAS6 Q14393 1/20 0.35
ALDH1A1 P00352 2/20 0.35
CYP19A1 P11511 1/20 0.34
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2910066 0.92 GSK3A (0.38) CDK1GSK3AGSK3BCD38AXL
SCHEMBL2909762 0.91 CDK1 (0.38) CDK1GSK3AGSK3BCD38ALDH1A1
SCHEMBL2903761 0.91 CDK1 (0.38) CDK1GSK3AGSK3BCD38ALDH1A1
SCHEMBL2911937 0.90 CDK1 (0.42) CDK1GSK3AGSK3BALDH1A1CYP19A1
SCHEMBL2909662 0.90 GSK3A (0.44) CDK1GSK3AGSK3BALDH1A1CYP19A1
SCHEMBL2904020 0.88 CDK1 (0.41) CDK1GSK3AGSK3BALDH1A1CYP19A1
SCHEMBL2904160 0.87 GSK3A (0.41) CDK1GSK3AGSK3BALDH1A1CYP19A1
SCHEMBL2903846 0.87 GSK3A (0.41) CDK1GSK3AGSK3BALDH1A1CYP19A1
SCHEMBL2904171 0.87 GSK3A (0.38) CDK1GSK3AGSK3BCD38AXL
SCHEMBL2911578 0.87 GSK3A (0.38) CDK1GSK3AGSK3BCD38AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed