SCHEMBL29133777

SCHEMBL29133777

COc1ncc(-c2ccc3ncnc(NCCc4ccccc4)c3c2)cc1NS(C)(=O)=O

nearest known ligand 0.75

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 14/20 0.75
PIK3CG P48736 4/20 0.68
PIK3CD O00329 3/20 0.68
PIK3CB P42338 3/20 0.68
EGFR P00533 3/20 0.65
PIK3R1 P27986 1/20 0.60
ALDH1A1 P00352 1/20 0.54
LMNA P02545 1/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CLK4 Q9HAZ1 1/20 0.54
PI4KA P42356 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29133751 0.88 EGFR (0.68) PIK3CAPIK3CGPIK3CDPIK3CBEGFR
SCHEMBL27170398 0.87 EGFR (0.84) PIK3CAPIK3CGPIK3CDPIK3CBEGFR
SCHEMBL29133727 0.85 PIK3CA (0.65) PIK3CAEGFRALDH1A1LMNACYP1A2
SCHEMBL29133708 0.83 EGFR (0.82) PIK3CAEGFRALDH1A1LMNACYP1A2
SCHEMBL24576803 0.82 PIK3CA (0.77) PIK3CAPIK3CGPIK3CDPIK3CBEGFR
SCHEMBL24576531 0.79 EGFR (1.00) PIK3CAPIK3CDEGFRALDH1A1LMNA
SCHEMBL27170399 0.79 EGFR (0.70) PIK3CAPIK3CGPIK3CDPIK3CBEGFR
SCHEMBL17845959 0.78 PIK3CA (0.66) PIK3CAPIK3CGPIK3CDPIK3CBEGFR
SCHEMBL29667014 0.78 PIK3CA (0.66) PIK3CAPIK3CGPIK3CDPIK3CBEGFR
SCHEMBL29133765 0.78 EGFR (0.54) PIK3CAPIK3CDEGFRPIK3R1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117295716-A Substituted aminobenzyl heteroaryl compounds as EGFR and/or PI3K inhibitors 麦克尼斯迪克治疗有限公司 2023-12-26 CN disclosed