SCHEMBL2913393

SCHEMBL2913393

CCOC(=O)c1cnc2cc(OCC)c(N3CCN(C(=O)OC(C)(C)C)CC3)cc2c1Nc1ccc(F)cc1F

nearest known ligand 0.68

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 10/20 0.68
KCNH2 Q12809 7/20 0.68
SCN5A Q14524 3/20 0.68
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2913106 0.97 KCNH2 (0.67) CSF1RKCNH2SCN5ALMNAMAPT
SCHEMBL2913425 0.95 CSF1R (0.64) CSF1RKCNH2SCN5AMAPT
SCHEMBL2904389 0.94 KCNH2 (0.69) CSF1RKCNH2SCN5ALMNAMAPT
SCHEMBL2911034 0.92 CSF1R (0.61) CSF1RKCNH2SCN5A
SCHEMBL2910312 0.90 KCNH2 (0.60) CSF1RKCNH2SCN5ALMNAMAPT
SCHEMBL2911029 0.89 CSF1R (0.84) CSF1RKCNH2SCN5A
SCHEMBL2911267 0.89 CSF1R (0.72) CSF1RKCNH2SCN5A
SCHEMBL2912345 0.88 CSF1R (0.71) CSF1RKCNH2SCN5ALMNAMAPT
SCHEMBL2914184 0.87 CSF1R (0.70) CSF1RKCNH2SCN5ALMNAMAPT
SCHEMBL2913777 0.87 KCNH2 (0.58) CSF1RKCNH2SCN5AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed