SCHEMBL29134305

SCHEMBL29134305

COC(=O)c1cnc(N2CCC(N(C)C(=O)OC(C)(C)C)C2)nc1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 1/20 0.48
PDE10A Q9Y233 2/20 0.45
HDAC6 Q9UBN7 1/20 0.43
JAK2 O60674 2/20 0.42
JAK3 P52333 2/20 0.42
GPR119 Q8TDV5 3/20 0.41
HSD11B1 P28845 1/20 0.41
VNN1 O95497 4/20 0.40
KDM4D Q6B0I6 1/20 0.39
SPR P35270 2/20 0.39
JAK1 P23458 1/20 0.39
USP30 Q70CQ3 2/20 0.38
OPRK1 P41145 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24033500 1.00 AAK1 (0.48) AAK1PDE10AHDAC6JAK2JAK3
SCHEMBL26712578 0.89 AAK1 (0.49) AAK1PDE10AHDAC6JAK2JAK3
SCHEMBL29134759 0.89 AAK1 (0.49) AAK1PDE10AHDAC6JAK2JAK3
Lithium Ion SCHEMBL30181681 0.87 AAK1 (0.46) AAK1PDE10AHDAC6JAK2JAK3
SCHEMBL2302835 0.85 AAK1 (0.48) AAK1PDE10AHDAC6JAK2JAK3
SCHEMBL2173915 0.85 AAK1 (0.48) AAK1PDE10AHDAC6JAK2JAK3
SCHEMBL24033406 0.83 AAK1 (0.48) AAK1PDE10AJAK2JAK3GPR119
SCHEMBL30665048 0.81 AAK1 (0.53) AAK1PDE10AJAK2JAK3GPR119
SCHEMBL24033388 0.81 AAK1 (0.53) AAK1PDE10AJAK2JAK3GPR119
SCHEMBL29134277 0.81 AAK1 (0.53) AAK1PDE10AJAK2JAK3GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116997548-A HTT modulators for the treatment of huntington's disease CHDI基金会股份有限公司 2023-11-03 CN disclosed