SCHEMBL29134491

SCHEMBL29134491

O=C(O)C1(c2ccc(Br)cc2)CSC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C1 Q04828 1/20 0.41
HDAC1 Q13547 3/20 0.37
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
OGG1 O15527 1/20 0.34
HDAC4 P56524 2/20 0.34
KMT2A Q03164 3/20 0.34
MEN1 O00255 2/20 0.34
TSHR P16473 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29134732 0.86 AKR1C1 (0.41) AKR1C1HDAC1ALDH1A1HDAC3HDAC7
SCHEMBL2221 0.82 AKR1C1 (0.55) AKR1C1HDAC1ALDH1A1KMT2AMEN1
SCHEMBL29134935 0.81 AKR1C1 (0.47) AKR1C1HDAC1ALDH1A1HDAC3HDAC7
SCHEMBL3910628 0.80 AKR1C1 (0.53) AKR1C1HDAC1ALDH1A1KMT2AMEN1
Water SCHEMBL3910626 0.78 AKR1C1 (0.52) AKR1C1HDAC1ALDH1A1KMT2AMEN1
SCHEMBL1492737 0.78 AKR1C1 (0.62) AKR1C1HDAC1ALDH1A1HDAC4KMT2A
SCHEMBL9966557 0.78 AKR1C1 (0.68) AKR1C1HDAC1ALDH1A1HDAC4KMT2A
SCHEMBL12988917 0.77 AKR1C1 (0.41) AKR1C1HDAC1CES2CES1ALDH1A1
Hydrochloric Acid SCHEMBL28915897 0.77 AKR1C1 (0.66) AKR1C1HDAC1ALDH1A1HDAC4KMT2A
SCHEMBL2384832 0.77 AKR1C1 (0.66) AKR1C1HDAC1ALDH1A1HDAC4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025137640-A1 AZASPIRO WRN INHIBITORS GILEAD SCIENCES, INC. (US) 2025-06-26 WO disclosed
EP-4313967-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-07 EP disclosed
CN-117120429-A KHK inhibitor 吉利德科学公司 2023-11-24 CN disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed