SCHEMBL29134660

SCHEMBL29134660

Cc1cc(-c2ccc(C#N)cc2)ccc1Nc1nc(Cl)ncc1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 2/20 0.45
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
TNIK Q9UKE5 2/20 0.39
HSD11B1 P28845 2/20 0.38
MAPKAPK2 P49137 2/20 0.37
KIF11 P52732 1/20 0.36
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
RIPK1 Q13546 1/20 0.36
AURKA O14965 1/20 0.35
LRRK2 Q5S007 1/20 0.35
P2RX7 Q99572 1/20 0.35
GSK3A P49840 1/20 0.35
GSK3B P49841 1/20 0.35
ALDH1A1 P00352 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PGR P06401 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30774987 1.00 SYK (0.45) SYKCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL30775005 0.90 SYK (0.48) SYKCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL29134663 0.90 SYK (0.48) SYKCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL29135024 0.87 CYP2C19 (0.48) SYKCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL30774992 0.87 CYP2C19 (0.48) SYKCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL29135028 0.85 CCNA2 (0.38) SYKCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL30774989 0.85 CCNA2 (0.38) SYKCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL30774990 0.81 CYP2C19 (0.50) SYKCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL29135023 0.81 CYP2C19 (0.50) SYKCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL15688460 0.78 SYK (0.72) SYKAURKAGSK3AGSK3BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117343017-A Halogenated diaryl pyrimidine compound containing biaryl structure, and preparation method and application thereof 四川大学 2024-01-05 CN disclosed