SCHEMBL2913657

SCHEMBL2913657

CC(C)(C)OC(=O)N1CC(O)CC1C(=O)Nc1cn(CCCNc2ccc([N+](=O)[O-])c(N)n2)cc1-c1ccc(Cl)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 4/20 0.44
GSK3A P49840 3/20 0.44
POLB P06746 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
ABL1 P00519 3/20 0.39
BCR P11274 3/20 0.39
CDK1 P06493 2/20 0.39
CCNB2 O95067 1/20 0.39
CCNB1 P14635 1/20 0.39
CCNB3 Q8WWL7 1/20 0.39
ALDH1A1 P00352 1/20 0.35
MCL1 Q07820 10/20 0.33
BCL2 P10415 2/20 0.33
BCL2L1 Q07817 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2910738 0.86 CYP1A2 (0.40) POLBCYP1A2CYP3A4CYP2C19ABL1
SCHEMBL2911302 0.82 GSK3B (0.47) GSK3BGSK3AABL1BCRCDK1
SCHEMBL2911295 0.82 GSK3B (0.47) GSK3BGSK3AABL1BCRCDK1
SCHEMBL2910561 0.81 GSK3B (0.51) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL1219461 0.81 GSK3B (0.49) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2911298 0.79 GSK3B (0.47) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2909927 0.79 GSK3B (0.49) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2910107 0.79 GSK3B (0.42) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2907714 0.78 GSK3B (0.42) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2904658 0.78 GSK3B (0.41) GSK3BGSK3ACDK1CCNB2CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed