SCHEMBL29136973

SCHEMBL29136973

Nc1nccc2cc(CCl)ccc12

nearest known ligand 0.72

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 14/20 0.72
ROCK2 O75116 1/20 0.54
KCNH2 Q12809 1/20 0.54
MAP4K4 O95819 1/20 0.50
F12 P00748 2/20 0.48
PLAU P00749 1/20 0.48
NCF1 P14598 1/20 0.48
NOS3 P29474 1/20 0.48
NOS1 P29475 1/20 0.48
NOS2 P35228 1/20 0.48
BACE1 P56817 1/20 0.48
KLKB1 P03952 4/20 0.46
KLK1 P06870 2/20 0.46
PLG P00747 1/20 0.44
F11 P03951 1/20 0.44
PRSS1 P07477 1/20 0.44
PRSS2 P07478 1/20 0.44
PRSS3 P35030 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5735425 0.84 ROCK1 (1.00) ROCK1ROCK2KCNH2MAP4K4F12
SCHEMBL29481418 0.84 ROCK1 (1.00) ROCK1ROCK2KCNH2MAP4K4F12
Hydrochloric Acid SCHEMBL29508477 0.82 ROCK1 (0.96) ROCK1ROCK2KCNH2MAP4K4F12
SCHEMBL28285945 0.82 ROCK1 (0.72) ROCK1ROCK2KCNH2MAP4K4F12
Hydrochloric Acid SCHEMBL29481411 0.82 ROCK1 (0.96) ROCK1ROCK2KCNH2MAP4K4F12
SCHEMBL1696126 0.82 ROCK1 (0.72) ROCK1ROCK2KCNH2MAP4K4F12
Hydrochloric Acid SCHEMBL3759590 0.82 ROCK1 (0.96) ROCK1ROCK2KCNH2MAP4K4F12
Hydrochloric Acid SCHEMBL5731184 0.82 ROCK1 (0.96) ROCK1ROCK2KCNH2MAP4K4F12
SCHEMBL22277251 0.79 ROCK1 (0.68) ROCK1ROCK2KCNH2MAP4K4F12
SCHEMBL13302588 0.78 ROCK1 (0.66) ROCK1ROCK2KCNH2MAP4K4F12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117355521-A Heteroaryl inhibitors of plasma kallikrein 武田药品工业株式会社 2024-01-05 CN disclosed