SCHEMBL29137574

SCHEMBL29137574

COc1cc(/C=C/C(=O)c2cc(OCc3ccccc3)cc(OCc3ccccc3)c2Br)ccc1OCc1ccccc1

nearest known ligand 0.73

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
APP P05067 10/20 0.61
PDE4A P27815 2/20 0.59
PDE4B Q07343 2/20 0.59
PDE4C Q08493 2/20 0.59
PDE4D Q08499 2/20 0.59
HPGD P15428 3/20 0.58
ALDH1A1 P00352 2/20 0.58
KDM4E B2RXH2 2/20 0.58
HTT P42858 1/20 0.58
GSK3B P49841 1/20 0.57
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
NPC1 O15118 1/20 0.53
MAPT P10636 1/20 0.53
RAB9A P51151 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2970084 0.88 APP (0.66) APPPDE4APDE4BPDE4CPDE4D
SCHEMBL19183186 0.82 PDE4A (0.70) APPPDE4APDE4BPDE4CPDE4D
SCHEMBL19183187 0.82 PDE4A (0.70) APPPDE4APDE4BPDE4CPDE4D
SCHEMBL30383293 0.82 MAOB (0.76) APPPDE4APDE4BPDE4CPDE4D
SCHEMBL10610437 0.82 PDE4A (0.74) APPPDE4APDE4BPDE4CPDE4D
SCHEMBL25214887 0.82 MAOB (0.76) APPPDE4APDE4BPDE4CPDE4D
SCHEMBL10610432 0.82 PDE4A (0.74) APPPDE4APDE4BPDE4CPDE4D
SCHEMBL25214886 0.82 MAOB (0.76) APPPDE4APDE4BPDE4CPDE4D
SCHEMBL31420038 0.82 NPC1 (0.78) APPPDE4APDE4BPDE4CPDE4D
SCHEMBL25265332 0.82 APP (0.78) APPHPGDALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113995738-B Application of 2' -halogenated chalcone derivative in preparation of medicine for treating liver related diseases 中国医学科学院药物研究所 2024-02-06 CN disclosed
CN-113979851-B 2' -halogenated chalcone derivative, preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2024-01-12 CN disclosed