SCHEMBL2914161

SCHEMBL2914161

CCCC(=O)Nc1ccc(C)c(-c2ccc(C(=O)O)cc2)c1

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 7/20 0.67
ALDH1A1 P00352 5/20 0.58
TP53 P04637 1/20 0.55
HPGD P15428 3/20 0.51
KDM4E B2RXH2 2/20 0.51
PTPRC P08575 2/20 0.50
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
HSD17B10 Q99714 1/20 0.48
F2R P25116 1/20 0.47
THRB P10828 1/20 0.47
MAPT P10636 1/20 0.47
FNTA P49354 1/20 0.46
FNTB P49356 1/20 0.46
RXRA P19793 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5028483 0.82 MAPK14 (0.58) MAPK14ALDH1A1TP53HPGDKDM4E
SCHEMBL2912882 0.82 MAPK14 (0.62) MAPK14ALDH1A1HPGDKDM4ECYP1A2
SCHEMBL2911571 0.82 MAPK14 (0.51) MAPK14RXRA
SCHEMBL2353921 0.81 LDLR (0.61) MAPK14ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL265614 0.81 TP53 (0.70) ALDH1A1TP53HPGDKDM4ECYP1A2
SCHEMBL2907534 0.81 MAPK14 (0.76) MAPK14
SCHEMBL2913317 0.81 MEN1 (0.59) MAPK14ALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL4813534 0.81 MAPK14 (1.00) MAPK14
SCHEMBL2912590 0.80 MAPK14 (0.50) MAPK14CYP1A2RXRA
SCHEMBL2912684 0.79 MAPK14 (0.69) MAPK14HPGDCYP1A2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940786-B1 BIPHENYL DERIVATIVES AND THEIR USE IN TREATING HEPATITIS C ARROW THERAPEUTICS LTD (GB) 2010-08-18 EP disclosed
US-20080255105-A1 Biphenyl Derivatives and Their Use in Treating Hepatitis C ARROW THERAPEUTICS LIMITED (GB) 2008-10-16 US disclosed
EP-1940786-A1 BIPHENYL DERIVATIVES AND THEIR USE IN TREATING HEPATITIS C Arrow Therapeutics Limited (GB) 2008-07-09 EP disclosed
WO-2007031791-A1 BIPHENYL DERIVATIVES AND THEIR USE IN TREATING HEPATITIS C ARROW THERAPEUTICS LIMITED (GB) 2007-03-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080255105-A1 Biphenyl Derivatives and Their Use in Treating Hepatitis C NR4A1, NR0B1, NR1H4 MAPK14 4315/4885ALDH1A1 441/4885TP53 1362/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.