SCHEMBL2915801

SCHEMBL2915801

[Pd].c1ccc(P(CCCP(c2ccccc2)c2ccccc2)c2ccccc2)cc1.c1ccc(P(CCCP(c2ccccc2)c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ESR1 P03372 4/20 0.33
ESR2 Q92731 4/20 0.33
KCNA3 P22001 1/20 0.31
CALM1 P0DP23 1/20 0.30
KDM4E B2RXH2 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4255002 1.00 CYP3A4 (0.43) CYP3A4TDP1ESR1ESR2KCNA3
Hydrochloric Acid SCHEMBL15253811 0.97 CYP3A4 (0.41) CYP3A4TDP1ESR1ESR2
Hydrochloric Acid SCHEMBL1025430 0.97 CYP3A4 (0.41) CYP3A4TDP1ESR1ESR2
SCHEMBL35092 0.97 CYP3A4 (0.45) CYP3A4TDP1ESR1ESR2KCNA3
SCHEMBL954340 0.94 CYP3A4 (0.43) CYP3A4TDP1ESR1ESR2KCNA3
SCHEMBL7934432 0.94 CYP3A4 (0.43) CYP3A4TDP1ESR1ESR2KCNA3
SCHEMBL556980 0.94 CYP3A4 (0.43) CYP3A4TDP1ESR1ESR2KCNA3
SCHEMBL22749132 0.94 CYP3A4 (0.43) CYP3A4TDP1ESR1ESR2KCNA3
SCHEMBL22749145 0.94 CYP3A4 (0.43) CYP3A4TDP1ESR1ESR2KCNA3
SCHEMBL31379074 0.94 CYP3A4 (0.43) CYP3A4TDP1ESR1ESR2KCNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653396-B1 Process for the preparation of 1,1'-binaphthylene HOECHST AG (DE) 1997-02-12 EP claimed
US-5510554-A REACTING A 1-HALO-2-SUBSTITUTED NAPHTHALENE WITH A 2-SUBSTITUTED-1-NAPHTHYL-MAGNESIUM HALIDE IN THE PRESENCE OF A PALLADIUM/PHOSPHINE CATALYST HOECHST AKTIENGESELLSCHAFT (DE) 1996-04-23 US claimed
EP-0653396-A1 Process for the preparation of 1,1'-binaphthylene HOECHST AKTIENGESELLSCHAFT (DE) 1995-05-17 EP claimed
US-8742127-B2 Production method of 6-halogeno-3-arylpyridine derivative KURARAY CO., LTD. (JP) 2014-06-03 US disclosed
US-20100280253-A1 PRODUCTION METHOD OF 6-HALOGENO-3-ARYLPYRIDINE DERIVATIVE KURARAY CO., LTD. (JP) 2010-11-04 US disclosed
EP-2223912-A1 METHOD FOR PRODUCING 6-HALOGENO-3-ARYLPYRIDINE DERIVATIVE Kuraray Co., Ltd. (JP) 2010-09-01 EP disclosed
EP-0653396-B1 Process for the preparation of 1,1'-binaphthylene HOECHST AG (DE) 1997-02-12 EP disclosed
EP-0743293-A1 Process for producing biaryl compound CHISSO CORPORATION (JP) 1996-11-20 EP disclosed
US-5510554-A REACTING A 1-HALO-2-SUBSTITUTED NAPHTHALENE WITH A 2-SUBSTITUTED-1-NAPHTHYL-MAGNESIUM HALIDE IN THE PRESENCE OF A PALLADIUM/PHOSPHINE CATALYST HOECHST AKTIENGESELLSCHAFT (DE) 1996-04-23 US disclosed
EP-0653396-A1 Process for the preparation of 1,1'-binaphthylene HOECHST AKTIENGESELLSCHAFT (DE) 1995-05-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100280253-A1 PRODUCTION METHOD OF 6-HALOGENO-3-ARYLPYRIDINE DERIVATIVE GMDS, MAP2, DDT CYP3A4 172/4885TDP1 1351/4885ESR1 4811/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.