SCHEMBL29171981

SCHEMBL29171981

Cc1nc2cc(-c3cc(C(=O)O)ccc3C(C)O)ccc2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.53
ESR2 Q92731 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
GRIK1 P39086 1/20 0.44
GRIA1 P42261 1/20 0.44
GRIA2 P42262 1/20 0.44
GRIA3 P42263 1/20 0.44
GRIA4 P48058 1/20 0.44
ALDH1A1 P00352 5/20 0.41
HPGD P15428 4/20 0.41
POLB P06746 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAPK1 P28482 1/20 0.39
TRPV1 Q8NER1 2/20 0.38
MLKL Q8NB16 2/20 0.37
KDM4E B2RXH2 3/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
DHODH Q02127 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30848269 1.00 HSP90AA1 (0.53) HSP90AA1ESR2TDP1GRIK1GRIA1
SCHEMBL30799117 0.90 CHEK2 (0.43) HSP90AA1ESR2TDP1CHEK2
SCHEMBL29172032 0.90 CHEK2 (0.43) HSP90AA1ESR2TDP1CHEK2
SCHEMBL30798800 0.88 TLR8 (0.43) HSP90AA1ESR2TDP1ALDH1A1HPGD
SCHEMBL29171974 0.88 BRD4 (0.48) HSP90AA1ESR2TDP1ALDH1A1HPGD
SCHEMBL30798804 0.83 TDP1 (0.58) HSP90AA1ESR2TDP1GRIK1GRIA1
SCHEMBL29171880 0.83 TDP1 (0.58) HSP90AA1ESR2TDP1GRIK1GRIA1
SCHEMBL29171943 0.82 BRD4 (0.47) POLBRAB9ASMN1; SMN2TRPV1BRD4
SCHEMBL30848037 0.82 BRD4 (0.47) POLBRAB9ASMN1; SMN2TRPV1BRD4
SCHEMBL30848167 0.80 HSP90AA1 (0.54) HSP90AA1ESR2TDP1GRIK1GRIA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117720472-A Benzimidazole compound, and preparation method and application thereof 苏州沪云新药研发股份有限公司 2024-03-19 CN disclosed