SCHEMBL29176302

SCHEMBL29176302

COc1ccc(-c2cc3c(cn2)n(C)c(=O)n3-c2cc(OC)c(OC)c(OC)c2)cc1O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KATNA1 O75449 1/20 0.52
MKNK2 Q9HBH9 1/20 0.41
TUBB4A P04350 5/20 0.41
TUBB P07437 5/20 0.41
TUBA3C P0DPH7 5/20 0.41
TUBA1B P68363 5/20 0.41
TUBA4A P68366 5/20 0.41
TUBB4B P68371 5/20 0.41
TUBB3 Q13509 5/20 0.41
TUBB2A Q13885 5/20 0.41
TUBB8 Q3ZCM7 5/20 0.41
TUBA3E Q6PEY2 5/20 0.41
TUBA1A Q71U36 5/20 0.41
TUBA1C Q9BQE3 5/20 0.41
TUBB6 Q9BUF5 5/20 0.41
TUBB2B Q9BVA1 5/20 0.41
TUBB1 Q9H4B7 5/20 0.41
PIK3CA P42336 1/20 0.39
MTOR P42345 1/20 0.39
PRKDC P78527 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30800001 1.00 KATNA1 (0.52) KATNA1MKNK2TUBB4ATUBBTUBA3C
SCHEMBL29176287 0.87 KATNA1 (0.50) KATNA1MKNK2TUBB4ATUBBTUBA3C
SCHEMBL30800071 0.87 KATNA1 (0.50) KATNA1MKNK2TUBB4ATUBBTUBA3C
SCHEMBL29176288 0.87 KATNA1 (0.50) KATNA1MKNK2TUBB4ATUBBTUBA3C
SCHEMBL28474690 0.85 KATNA1 (0.49) KATNA1MKNK2TUBB4ATUBBTUBA3C
SCHEMBL30799997 0.84 KATNA1 (0.54) KATNA1MKNK2TUBB4ATUBBTUBA3C
SCHEMBL29176273 0.84 KATNA1 (0.54) KATNA1MKNK2TUBB4ATUBBTUBA3C
SCHEMBL29176281 0.80 KATNA1 (0.64) KATNA1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL30800023 0.80 KATNA1 (0.64) KATNA1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL30799979 0.70 BLK (0.46) KATNA1TUBB4ATUBBTUBA3CTUBA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111732584-B Diaryl substituted fused heterocycle compound and preparation method and application thereof in pharmacy 复旦大学 2024-02-27 CN disclosed