SCHEMBL2919259

SCHEMBL2919259

C/C=C(/F)COc1ccc2sc(-c3ccc(C)cc3)nc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 8/20 0.48
MAPT P10636 6/20 0.48
TP53 P04637 5/20 0.48
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.45
THRB P10828 2/20 0.45
RXFP1 Q9HBX9 1/20 0.44
DYRK1A Q13627 3/20 0.44
KDM4E B2RXH2 3/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
ALDH1A1 P00352 2/20 0.43
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
HTT P42858 1/20 0.43
HDAC6 Q9UBN7 1/20 0.42
APP P05067 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2923395 0.91 MAPT (0.52) SMN1; SMN2MAPTTP53LMNAPOLB
SCHEMBL3757505 0.89 AOC3 (0.47) SMN1; SMN2MAPTTP53LMNAPOLB
SCHEMBL3757503 0.89 AOC3 (0.47) SMN1; SMN2MAPTTP53LMNAPOLB
SCHEMBL3757500 0.89 AOC3 (0.47) SMN1; SMN2MAPTTP53LMNAPOLB
Hydrochloric Acid SCHEMBL3757804 0.88 AOC3 (0.46) SMN1; SMN2MAPTTP53LMNAPOLB
Hydrochloric Acid SCHEMBL3757799 0.88 AOC3 (0.46) SMN1; SMN2MAPTTP53LMNAPOLB
Hydrochloric Acid SCHEMBL3757801 0.88 AOC3 (0.46) SMN1; SMN2MAPTTP53LMNAPOLB
SCHEMBL3751571 0.83 PDE10A (0.51) SMN1; SMN2MAPTTP53LMNAPOLB
SCHEMBL3751570 0.83 PDE10A (0.51) SMN1; SMN2MAPTTP53LMNAPOLB
SCHEMBL2940590 0.80 MAPT (0.48) SMN1; SMN2MAPTTP53THRBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222160-A2 HALOALLYLAMINE INHIBITORS OF SSAO/VAP-1 AND USES THEREFOR Pharmaxis Ltd. (AU) 2010-09-01 EP claimed
WO-2009066152-A2 HALOALLYLAMINE INHIBITORS OF SSAO/VAP-1 AND USES THEREFOR PHARMAXIS LTD. (US) 2009-05-28 WO claimed