SCHEMBL2919558

SCHEMBL2919558

Cc1c(F)ccc2cnc(Nc3cc(N)c4cn[nH]c4c3)nc12

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 2/20 0.40
SYK P43405 9/20 0.39
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
PDGFRB P09619 4/20 0.35
PDGFRA P16234 4/20 0.35
IGF1R P08069 1/20 0.34
BTK Q06187 2/20 0.34
LYN P07948 1/20 0.34
TXK P42681 1/20 0.34
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34
JAK3 P52333 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2919211 0.89 CDC7 (0.41) CDC7SYKPDGFRBPDGFRAIGF1R
SCHEMBL2918438 0.85 IGF1R (0.46) CDC7SYKPDGFRBPDGFRAIGF1R
SCHEMBL2919831 0.85 IGF1R (0.43) SYKPDGFRBPDGFRAIGF1RJAK2
SCHEMBL2918594 0.83 CDC7 (0.58) CDC7SYKPDGFRBPDGFRAIGF1R
SCHEMBL2920288 0.83 PDGFRB (0.37) CDC7SYKPDGFRBPDGFRAIGF1R
SCHEMBL2921534 0.83 SYK (0.41) SYKIDO1TDO2BTKLYN
SCHEMBL2918740 0.82 CDK1 (0.42) SYKJAK2JAK1TYK2JAK3
SCHEMBL2916296 0.81 TTK (0.35) CDC7SYKIDO1TDO2PDGFRB
SCHEMBL2918651 0.79 KIT (0.38) CDC7SYKIDO1TDO2BTK
SCHEMBL2919791 0.78 SYK (0.41) CDC7SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100311965-A1 2-AMINOQUINAZOLINE DERIVATIVE CARNA BIOSCIENCES INC. (JP) 2010-12-09 US disclosed
US-20100311965-A1 2-AMINOQUINAZOLINE DERIVATIVE CARNA BIOSCIENCES INC. (JP) 2010-12-09 US disclosed
US-20100311965-A1 2-AMINOQUINAZOLINE DERIVATIVE CARNA BIOSCIENCES INC. (JP) 2010-12-09 US disclosed
EP-2226315-A1 2-AMINOQUINAZOLINE DERIVATIVE Carna Biosciences Inc. (JP) 2010-09-08 EP disclosed
WO-2009084695-A1 2-AMINOQUINAZOLINE DERIVATIVE CARNA BIOSCIENCES INC. (JP) 2009-07-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100311965-A1 2-AMINOQUINAZOLINE DERIVATIVE DSTYK, ABL1, EEF2K CDC7 405/4885SYK 724/4885IDO1 2664/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.