SCHEMBL29201164

SCHEMBL29201164

CCOC(=O)C(c1ccccc1)C(c1ccc([N+](=O)[O-])cc1)c1cccc2c1CCN(c1ccc([N+](=O)[O-])cc1)C2

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
MAPT P10636 8/20 0.44
ALDH1A1 P00352 6/20 0.44
LMNA P02545 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
HTR1A P08908 1/20 0.39
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
HTT P42858 1/20 0.38
AR P10275 1/20 0.37
GAA P10253 1/20 0.37
POLB P06746 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
TP53 P04637 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29201153 0.95 MEN1 (0.43) MEN1KMT2AMAPTALDH1A1LMNA
SCHEMBL28739004 0.87 ACACB (0.45) MEN1KMT2AMAPTALDH1A1LMNA
SCHEMBL28940362 0.87 HPGD (0.49) MEN1KMT2AMAPTALDH1A1LMNA
SCHEMBL28739260 0.87 HPGD (0.52) MEN1KMT2AALDH1A1SMN1; SMN2HTT
SCHEMBL28739124 0.87 ACACB (0.47) ALDH1A1
SCHEMBL30768144 0.84 MEN1 (0.48) MEN1KMT2AMAPTALDH1A1LMNA
SCHEMBL29201149 0.84 MEN1 (0.48) MEN1KMT2AMAPTALDH1A1LMNA
SCHEMBL28739075 0.83 ACACB (0.43)
SCHEMBL28739086 0.83 HPGD (0.47) MEN1KMT2AMAPTALDH1A1LMNA
SCHEMBL28739100 0.83 ACACB (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114507181-B Propionic acid compound containing 5-substituted tetrahydroisoquinoline, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2024-03-26 CN disclosed