SCHEMBL29212657

SCHEMBL29212657

CCN(CC)c1nc2ccc(-c3nc(NC4CCN(S(C)(=O)=O)CC4)ncc3F)cc2s1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DYRK2 Q92630 11/20 0.58
CCNE1 P24864 5/20 0.56
CDK2 P24941 5/20 0.56
CDK1 P06493 3/20 0.56
CCNB1 P14635 3/20 0.56
CCNB2 O95067 2/20 0.56
CCNE2 O96020 2/20 0.56
CDK5 Q00535 2/20 0.56
CDK5R1 Q15078 2/20 0.56
CCNB3 Q8WWL7 2/20 0.56
CDK6 Q00534 5/20 0.48
CDK4 P11802 4/20 0.48
CCND1 P24385 4/20 0.48
CCND3 P30281 4/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29212666 0.87 DYRK2 (0.71) DYRK2CDK6
SCHEMBL29212669 0.84 DYRK2 (0.72) DYRK2CCNE1CDK2CDK1CCNB1
SCHEMBL31472289 0.84 CDK2 (0.58) DYRK2CCNE1CDK2CDK1CCNB1
SCHEMBL29233639 0.84 CDK2 (0.58) DYRK2CCNE1CDK2CDK1CCNB1
SCHEMBL30883983 0.82 DYRK2 (0.64) DYRK2CCNE1CDK2CDK1CCNB1
SCHEMBL29212665 0.82 DYRK2 (0.64) DYRK2CCNE1CDK2CDK1CCNB1
SCHEMBL30569710 0.81 DYRK2 (0.74) DYRK2CDK6CDK4CCND1CCND3
SCHEMBL26451650 0.81 DYRK2 (0.74) DYRK2CDK6CDK4CCND1CCND3
SCHEMBL31472288 0.80 CDK2 (0.66) DYRK2CCNE1CDK2CDK1CCNB1
SCHEMBL29233646 0.80 CDK2 (0.66) DYRK2CCNE1CDK2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118005624-A Pyrimidine benzo five-membered ring CDK inhibitor and preparation method and application thereof 中国药科大学 2024-05-10 CN disclosed