SCHEMBL29216896

SCHEMBL29216896

Cc1cccc(F)c1C(=O)Nc1cnc(-c2ccc(Br)cc2Cl)cn1

nearest known ligand 0.69

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
STIM1 Q13586 1/20 0.69
ORAI1 Q96D31 1/20 0.69
ORAI2 Q96SN7 1/20 0.69
IL2 P60568 15/20 0.52
L3MBTL1 Q9Y468 1/20 0.44
PTGFR P43088 1/20 0.41
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
MAPK1 P28482 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15395777 0.86 STIM1 (0.63) STIM1ORAI1ORAI2IL2L3MBTL1
Zegocractin SCHEMBL29391484 0.82 STIM1 (1.00) STIM1ORAI1ORAI2IL2L3MBTL1
Zegocractin SCHEMBL29362538 0.82 STIM1 (1.00) STIM1ORAI1ORAI2IL2L3MBTL1
Zegocractin SCHEMBL18038390 0.82 STIM1 (1.00) STIM1ORAI1ORAI2IL2L3MBTL1
SCHEMBL29216902 0.81 STIM1 (0.60) STIM1ORAI1ORAI2IL2L3MBTL1
SCHEMBL8260054 0.80 STIM1 (0.67) STIM1ORAI1ORAI2IL2L3MBTL1
SCHEMBL17244766 0.80 STIM1 (0.69) STIM1ORAI1ORAI2IL2L3MBTL1
SCHEMBL15395969 0.80 STIM1 (0.58) STIM1ORAI1ORAI2IL2L3MBTL1
SCHEMBL5554192 0.79 STIM1 (0.57) STIM1ORAI1ORAI2IL2L3MBTL1
SCHEMBL5555312 0.79 STIM1 (0.57) STIM1ORAI1ORAI2IL2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118084860-A Aromatic amide compound, pharmaceutical composition and application thereof 中国药科大学 2024-05-28 CN disclosed