SCHEMBL2922682

SCHEMBL2922682

Cc1c(N2CCC(CCO)CC2)ccc2cnc(Nc3ccc4cn[nH]c4c3)nc12

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 12/20 0.48
PDGFRA P16234 12/20 0.48
EGFR P00533 1/20 0.43
FGFR1 P11362 1/20 0.43
JAK3 P52333 1/20 0.43
SYK P43405 3/20 0.43
CDK4 P11802 2/20 0.42
CCND1 P24385 2/20 0.42
CDK1 P06493 1/20 0.42
CCNB1 P14635 1/20 0.42
CCNE1 P24864 1/20 0.42
CDK2 P24941 1/20 0.42
CDC7 O00311 1/20 0.41
WEE1 P30291 1/20 0.41
CCND2 P30279 1/20 0.41
CCND3 P30281 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2917783 0.93 PDGFRB (0.49) PDGFRBPDGFRAEGFRFGFR1JAK3
SCHEMBL2921459 0.85 PDGFRB (0.54) PDGFRBPDGFRAEGFRFGFR1SYK
SCHEMBL2921831 0.84 PDGFRB (0.54) PDGFRBPDGFRAEGFRFGFR1SYK
SCHEMBL2917218 0.84 PDGFRB (0.63) PDGFRBPDGFRAEGFRFGFR1CDK4
SCHEMBL2911263 0.84 PDGFRB (0.65) PDGFRBPDGFRAEGFRFGFR1JAK3
SCHEMBL2912670 0.83 PDGFRB (0.65) PDGFRBPDGFRAEGFRFGFR1SYK
SCHEMBL2921103 0.82 PDGFRB (0.41) PDGFRBPDGFRAJAK3CDK4CCND1
SCHEMBL2912102 0.81 SYK (0.61) PDGFRBPDGFRAEGFRFGFR1JAK3
SCHEMBL2913098 0.81 CDK4 (0.42) PDGFRBPDGFRAJAK3CDK4CCND1
SCHEMBL2917536 0.81 CDK1 (0.39) PDGFRBPDGFRAJAK3SYKCDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100311965-A1 2-AMINOQUINAZOLINE DERIVATIVE CARNA BIOSCIENCES INC. (JP) 2010-12-09 US disclosed
US-20100311965-A1 2-AMINOQUINAZOLINE DERIVATIVE CARNA BIOSCIENCES INC. (JP) 2010-12-09 US disclosed
US-20100311965-A1 2-AMINOQUINAZOLINE DERIVATIVE CARNA BIOSCIENCES INC. (JP) 2010-12-09 US disclosed
EP-2226315-A1 2-AMINOQUINAZOLINE DERIVATIVE Carna Biosciences Inc. (JP) 2010-09-08 EP disclosed
EP-2226315-A1 2-AMINOQUINAZOLINE DERIVATIVE Carna Biosciences Inc. (JP) 2010-09-08 EP disclosed
WO-2009084695-A1 2-AMINOQUINAZOLINE DERIVATIVE CARNA BIOSCIENCES INC. (JP) 2009-07-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100311965-A1 2-AMINOQUINAZOLINE DERIVATIVE DSTYK, ABL1, EEF2K PDGFRB 1018/4885PDGFRA 862/4885EGFR 479/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.