SCHEMBL29227197

SCHEMBL29227197

COc1ccc2ccccc2c1C=NNC(=O)CCc1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.62
CYP1A2 P05177 1/20 0.62
CYP3A4 P08684 1/20 0.62
CYP2C9 P11712 1/20 0.62
CYP2C19 P33261 1/20 0.62
ALDH1A1 P00352 5/20 0.60
KDM4E B2RXH2 6/20 0.59
HPGD P15428 4/20 0.59
GAA P10253 3/20 0.59
HTT P42858 1/20 0.59
POLB P06746 2/20 0.58
KMT2A Q03164 7/20 0.57
NPC1 O15118 4/20 0.57
MEN1 O00255 6/20 0.56
USP2 O75604 1/20 0.55
IDO1 P14902 2/20 0.55
ATM Q13315 1/20 0.55
RAB9A P51151 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13628768 0.81 SGK1 (0.64) MAPTALDH1A1KDM4EHPGDGAA
SCHEMBL24175846 0.80 MEN1 (0.78) MAPTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL14642552 0.76 HPGD (0.55) MAPTALDH1A1KDM4EHPGDGAA
SCHEMBL16993698 0.76 KDM4E (0.63) MAPTALDH1A1KDM4EHPGDGAA
SCHEMBL16993697 0.76 KDM4E (0.63) MAPTALDH1A1KDM4EHPGDGAA
Hydrochloric Acid SCHEMBL6510818 0.75 KDM4E (0.62) MAPTALDH1A1KDM4EHPGDGAA
Hydrochloric Acid SCHEMBL6510823 0.75 KDM4E (0.62) MAPTALDH1A1KDM4EHPGDGAA
SCHEMBL13954727 0.75 MAPT (0.67) MAPTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6494638 0.74 POLB (0.78) MAPTALDH1A1KDM4EGAAPOLB
SCHEMBL14642553 0.74 HPGD (0.51) MAPTALDH1A1KDM4EHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117946031-A Substituted aromatic phenol derivatives of KNa1.1 channel inhibitors 北京大学 2024-04-30 CN disclosed