SCHEMBL29236199

SCHEMBL29236199

O=C(Nc1ccc(F)cn1)c1cc(Br)cc(F)c1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.47
SORT1 Q99523 2/20 0.47
NPC1 O15118 4/20 0.45
RAB9A P51151 4/20 0.45
TP53 P04637 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 1/20 0.45
GLA P06280 1/20 0.45
GAA P10253 1/20 0.45
HSD17B10 Q99714 1/20 0.45
MAPK1 P28482 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
GRM5 P41594 3/20 0.44
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 1/20 0.43
SLC6A3 Q01959 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31027173 1.00 AHR (0.47) AHRSORT1NPC1RAB9ATP53
SCHEMBL31027174 1.00 AHR (0.47) AHRSORT1NPC1RAB9ATP53
SCHEMBL3851843 0.85 NPC1 (0.57) AHRSORT1NPC1RAB9ATP53
SCHEMBL29236313 0.79 CYP3A4 (0.49) AHRGRM5CYP1A2CYP3A4SLC6A3
SCHEMBL30300325 0.79 CYP3A4 (0.49) AHRGRM5CYP1A2CYP3A4SLC6A3
SCHEMBL3852931 0.77 NPC1 (0.60) AHRSORT1NPC1RAB9ATP53
SCHEMBL20177030 0.76 KDM4E (0.64) NPC1RAB9ATP53SMN1; SMN2KDM4E
SCHEMBL21579395 0.76 NPC1 (0.50) NPC1RAB9ATP53KDM4EMAPK1
SCHEMBL29236270 0.75 GRM5 (0.44) AHRNPC1RAB9ATP53SMN1; SMN2
SCHEMBL29236307 0.74 AHR (0.47) AHRNPC1RAB9AMAPK1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118234718-A Phenyl core compounds as MGLU5 negative allosteric modulators and methods of making and using the same 范德比尔特大学 2024-06-21 CN disclosed