SCHEMBL2923992

SCHEMBL2923992

COC(=O)c1cccc(Nc2c(-c3ccccc3)nc3cnccn23)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SALL4 Q9UJQ4 1/20 0.71
SYK P43405 1/20 0.69
GAA P10253 11/20 0.61
KDM4E B2RXH2 6/20 0.61
LMNA P02545 3/20 0.61
MAPK1 P28482 2/20 0.61
MAPT P10636 9/20 0.60
ALDH1A1 P00352 5/20 0.60
HSD17B10 Q99714 2/20 0.60
MEN1 O00255 1/20 0.60
KMT2A Q03164 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
BRAF P15056 3/20 0.58
TUBB4A P04350 2/20 0.55
TUBB P07437 2/20 0.55
TUBA3C P0DPH7 2/20 0.55
TUBA1B P68363 2/20 0.55
TUBA4A P68366 2/20 0.55
TUBB4B P68371 2/20 0.55
TUBB3 Q13509 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31355261 1.00 SALL4 (0.71) SALL4SYKGAAKDM4ELMNA
SCHEMBL31355335 0.94 SALL4 (0.69) SALL4SYKGAAKDM4ELMNA
SCHEMBL31355390 0.91 SYK (0.81) SALL4SYKGAAKDM4ELMNA
SCHEMBL31355339 0.90 SYK (0.85) SALL4SYKGAAKDM4ELMNA
SCHEMBL31355280 0.90 GAA (0.67) SALL4SYKGAAKDM4ELMNA
SCHEMBL26908187 0.89 GAA (0.71) SALL4SYKGAAKDM4ELMNA
SCHEMBL31355374 0.88 SYK (0.69) SALL4SYKGAAKDM4ELMNA
SCHEMBL31355274 0.87 SYK (0.66) SALL4SYKGAAKDM4ELMNA
SCHEMBL31355404 0.86 MAPT (0.77) SALL4SYKGAAKDM4ELMNA
SCHEMBL29818731 0.86 GAA (0.64) SALL4SYKGAAKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1901748-B1 ANGIOGENESIS INHIBITORS ONCALIS AG (CH) 2010-09-08 EP disclosed
EP-1901748-B1 ANGIOGENESIS INHIBITORS ONCALIS AG (CH) 2010-09-08 EP disclosed
EP-1765351-B9 PROTEIN KINASE INHIBITORS ONCALIS AG (CH) 2010-03-24 EP disclosed
EP-1765351-B9 PROTEIN KINASE INHIBITORS ONCALIS AG (CH) 2010-03-24 EP disclosed
EP-1765351-B1 PROTEIN KINASE INHIBITORS ONCALIS AG (CH) 2009-03-04 EP disclosed
EP-1765351-B1 PROTEIN KINASE INHIBITORS ONCALIS AG (CH) 2009-03-04 EP disclosed
US-20070149535-A1 Protein kinase inhibitors ONCALIS AG (CH) 2007-06-28 US disclosed
US-20070149535-A1 Protein kinase inhibitors ONCALIS AG (CH) 2007-06-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070149535-A1 Protein kinase inhibitors FLT1, ERBB2, ERBB3 SALL4 2422/4885SYK 469/4885GAA 3677/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.