SCHEMBL29256708

SCHEMBL29256708

Cc1nc(N2CCCCCC2)c(C(=O)Nc2cccc(C#N)c2)cc1Cl

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 8/20 0.55
TP53 P04637 2/20 0.51
P2RX1 P51575 1/20 0.48
ALDH1A1 P00352 2/20 0.47
HTT P42858 1/20 0.47
GRM4 Q14833 1/20 0.46
LMNA P02545 1/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
MAPK1 P28482 1/20 0.45
KMT2A Q03164 1/20 0.45
EPAS1 Q99814 1/20 0.45
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29256608 1.00 SCN10A (0.55) SCN10ATP53P2RX1ALDH1A1HTT
SCHEMBL29256631 0.99 SCN10A (0.54) SCN10ATP53P2RX1ALDH1A1HTT
SCHEMBL29256576 0.90 PPARG (0.54) SCN10AP2RX1ALDH1A1HTTKDM4E
SCHEMBL29256581 0.89 SCN10A (0.64) SCN10A
SCHEMBL29256616 0.85 SCN10A (0.67) SCN10ATP53P2RX1HTTGRM4
SCHEMBL29256590 0.85 SCN10A (0.67) SCN10ATP53P2RX1HTTGRM4
SCHEMBL31037390 0.85 SCN10A (0.67) SCN10ATP53P2RX1HTTGRM4
SCHEMBL31037437 0.84 SCN10A (0.66) SCN10ATP53P2RX1HTTGRM4
SCHEMBL29256637 0.84 SCN10A (0.66) SCN10ATP53P2RX1HTTGRM4
SCHEMBL23779638 0.82 SCN10A (0.82) SCN10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024217344-A1 NAV1.8 INHIBITORS, PREPARATION METHOD THEREFOR AND USE THEREOF 中国科学院上海药物研究所 2024-10-24 WO disclosed
CN-118324743-A Nav1.8 inhibitor and preparation method and application thereof 中国科学院上海药物研究所 2024-07-12 CN disclosed