SCHEMBL29258458

SCHEMBL29258458

Cc1nc(N2CCC(C(=O)NS(=O)(=O)c3ccc(Cl)s3)C2)c(C#N)cc1C(=O)O

nearest known ligand 0.74

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 19/20 0.74
CYP3A4 P08684 2/20 0.60
CYP2C9 P11712 2/20 0.60
CYP1A2 P05177 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C19 P33261 1/20 0.60
CHRM2 P08172 1/20 0.49
DRD3 P35462 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4109942 0.95 P2RY12 (0.81) P2RY12CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL29258649 0.93 P2RY12 (0.81) P2RY12CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL29258436 0.90 P2RY12 (0.91) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL4099779 0.89 P2RY12 (0.82) P2RY12CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL29258452 0.88 P2RY12 (0.80) P2RY12CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL29258457 0.87 P2RY12 (0.79) P2RY12CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL5315088 0.86 P2RY12 (0.69) P2RY12CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL4098046 0.85 P2RY12 (1.00) P2RY12CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL29258845 0.84 P2RY12 (0.73) P2RY12CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL4097423 0.83 P2RY12 (1.00) P2RY12CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118344351-A Preparation method and application of PET imaging agent targeting neuroinflammatory purinergic P2Y12 receptor 复旦大学 2024-07-16 CN disclosed