SCHEMBL2925964

SCHEMBL2925964

COc1cccc2cc(C3CCNCC3)c(=O)[nH]c12

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 4/20 0.54
BRD4 O60885 3/20 0.44
ATAD2 Q6PL18 3/20 0.44
HTR1A P08908 2/20 0.43
SLC6A2 P23975 2/20 0.43
SLC6A4 P31645 2/20 0.43
SLC6A3 Q01959 2/20 0.43
HTR6 P50406 4/20 0.42
JUND P17535 1/20 0.41
FOSB P53539 1/20 0.41
BRPF1 P55201 1/20 0.41
HRH4 Q9H3N8 1/20 0.41
PLAT P00750 1/20 0.40
CDK1 P06493 1/20 0.40
CDK9 P50750 1/20 0.40
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3543444 0.80 DAO (0.52) HTR2CBRD4ATAD2HTR1ASLC6A2
SCHEMBL13792219 0.80 DAO (0.52) HTR2CBRD4ATAD2HTR1ASLC6A2
Hydrochloric Acid SCHEMBL2211935 0.79 DAO (0.51) HTR2CBRD4ATAD2HTR1ASLC6A2
Hydrochloric Acid SCHEMBL2212880 0.79 DAO (0.51) HTR2CBRD4ATAD2HTR1ASLC6A2
Acetic Acid SCHEMBL3891621 0.77 DAO (0.49) BRD4ATAD2HTR1ASLC6A2SLC6A4
SCHEMBL27696635 0.75 HTR2C (0.66) HTR2CHTR1ASLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL3894574 0.74 HTR2C (0.67) HTR2CHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL105569 0.74 MAOB (0.48) HTR2CBRD4HRH4
SCHEMBL2260023 0.73 KDM4E (0.51) HTR2CHTR6
Hydrochloric Acid SCHEMBL31318331 0.72 HTR2C (0.48) HTR2CBRD4HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225223-B1 ORGANIC COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2017-01-11 EP disclosed
EP-2205590-B1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2014-06-04 EP disclosed
EP-2251338-A2 Organic compounds Boehringer Ingelheim International GmbH (DE) 2010-11-17 EP disclosed
EP-2225223-A2 ORGANIC COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2010-09-08 EP disclosed
EP-2205590-A1 CGRP ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2010-07-14 EP disclosed
WO-2009065919-A2 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-05-28 WO disclosed
WO-2009050232-A1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-04-23 WO disclosed