SCHEMBL2925982

SCHEMBL2925982

Nc1ccccc1Cc1cccc2nc(N[C@@H]3CCc4ccccc43)ccc12

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 2/20 0.41
PDPK1 O15530 1/20 0.40
JAK2 O60674 3/20 0.39
JAK3 P52333 3/20 0.39
FADS1 O60427 1/20 0.39
PARP1 P09874 2/20 0.38
HDAC6 Q9UBN7 1/20 0.38
KCNN3 Q9UGI6 1/20 0.38
AURKA O14965 1/20 0.37
RPS6KB1 P23443 1/20 0.37
PFKFB3 Q16875 1/20 0.37
EGFR P00533 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1615946 0.89 GBA1 (0.48) GBA1PDPK1JAK2JAK3FADS1
SCHEMBL1615945 0.89 GBA1 (0.48) GBA1PDPK1JAK2JAK3FADS1
SCHEMBL1615788 0.86 GBA1 (0.44) GBA1PDPK1JAK2JAK3FADS1
SCHEMBL2245619 0.81 GBA1 (0.47) GBA1PDPK1FADS1PARP1HDAC6
SCHEMBL3844986 0.80 PDPK1 (0.47) GBA1PDPK1JAK2JAK3FADS1
SCHEMBL1616344 0.79 GBA1 (0.46) GBA1PDPK1JAK2JAK3FADS1
SCHEMBL1616343 0.79 GBA1 (0.46) GBA1PDPK1JAK2JAK3FADS1
SCHEMBL1616249 0.78 GBA1 (0.50) GBA1PDPK1FADS1PARP1HDAC6
SCHEMBL1616241 0.78 GBA1 (0.50) GBA1PDPK1FADS1PARP1HDAC6
SCHEMBL1616604 0.76 GBA1 (0.43) GBA1PDPK1FADS1PARP1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099763-B1 2-AMINOQUINOLINES AS 5-HT(5A) RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed