SCHEMBL29277692

SCHEMBL29277692

COC(=O)c1nc(OBO)cnc1NC(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.39
MAPKAPK2 P49137 5/20 0.34
GSK3B P49841 1/20 0.34
DYRK1A Q13627 1/20 0.34
NPSR1 Q6W5P4 2/20 0.33
ACVR1B P36896 1/20 0.33
TGFBR1 P36897 1/20 0.33
ACVRL1 P37023 1/20 0.33
STK17B O94768 1/20 0.32
STK17A Q9UEE5 1/20 0.32
SYK P43405 2/20 0.32
LCK P06239 1/20 0.31
METAP1 P53582 1/20 0.31
NAMPT P43490 1/20 0.31
PRMT1 Q99873 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29277697 0.81 ATR (0.49) ATRMAPKAPK2GSK3BDYRK1ANPSR1
SCHEMBL7462692 0.80 ATR (0.42) ATRMAPKAPK2GSK3BDYRK1ANPSR1
SCHEMBL7455428 0.79 ATR (0.41) ATRMAPKAPK2GSK3BDYRK1ANPSR1
SCHEMBL29277701 0.78 ATR (0.41) ATRMAPKAPK2GSK3BDYRK1ANPSR1
SCHEMBL15402213 0.76 MAPKAPK2 (0.47) ATRMAPKAPK2
SCHEMBL29277699 0.74 NPSR1 (0.41) ATRDYRK1ANPSR1
SCHEMBL9897763 0.71 ATR (0.39) ATRMAPKAPK2GSK3BDYRK1ANPSR1
SCHEMBL32681564 0.70 SYK (0.39) ATRMAPKAPK2GSK3BDYRK1ANPSR1
SCHEMBL25138307 0.69 ATR (0.42) ATRACVR1BTGFBR1ACVRL1SYK
SCHEMBL12233051 0.69 MAPKAPK2 (0.44) ATRMAPKAPK2GSK3BDYRK1ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117327053-A Preparation method of PKC inhibitor darovasertib 云南万宏医药科技有限公司 2024-01-02 CN disclosed