SCHEMBL29281024

SCHEMBL29281024

Cc1onc(C(N)=O)c1F

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39
GRIA1 P42261 1/20 0.38
GRIA3 P42263 1/20 0.38
POLB P06746 2/20 0.37
TSHR P16473 2/20 0.37
HSD17B10 Q99714 1/20 0.35
ALDH1A1 P00352 2/20 0.32
HTT P42858 2/20 0.32
AR P10275 1/20 0.32
LMNA P02545 1/20 0.31
RECQL P46063 1/20 0.31
IKBKB O14920 1/20 0.31
HCAR2 Q8TDS4 1/20 0.31
GPX4 P36969 1/20 0.30
BTK Q06187 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31226280 0.79 MAPT (0.44) GAAGRIA1GRIA3POLBTSHR
SCHEMBL2676823 0.78 MEN1 (0.41) MEN1GAAKMT2AGRIA1GRIA3
SCHEMBL31226160 0.76 NPSR1 (0.45) MEN1KMT2APOLBHSD17B10ALDH1A1
SCHEMBL3189125 0.75 TSHR (0.44) MEN1GAAKMT2AGRIA1GRIA3
SCHEMBL3170099 0.72 GRIA1 (0.46) MEN1GAAKMT2AGRIA1GRIA3
SCHEMBL31301207 0.70 POLB (0.34) MEN1GAAKMT2AGRIA1GRIA3
SCHEMBL3179817 0.69 GRIA1 (0.44) MEN1GAAKMT2AGRIA1GRIA3
SCHEMBL18742872 0.69
SCHEMBL3175473 0.68 GRIA1 (0.54) MEN1GAAKMT2AGRIA1GRIA3
SCHEMBL15652402 0.68 GRIA1 (0.43) MEN1GAAKMT2AGRIA1GRIA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118546134-A Crystal form containing aromatic ring derivative antagonist, preparation method and application thereof 江苏豪森药业集团有限公司 2024-08-27 CN disclosed
CN-117836294-A Biological antagonist containing aromatic ring, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-04-05 CN disclosed