SCHEMBL292923

SCHEMBL292923

NC1CCN(c2nc(NCC(c3ccccc3)c3ccccc3)c3ncn([C@@H]4C[C@H](NC(=O)CO)[C@@H](O)[C@H]4O)c3n2)C1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 15/20 0.54
ADORA3 P0DMS8 7/20 0.54
CCNE2 O96020 1/20 0.44
CCNA2 P20248 1/20 0.44
CCNE1 P24864 1/20 0.44
CDK2 P24941 1/20 0.44
CCNA1 P78396 1/20 0.44
ADORA2B P29275 1/20 0.42
ADORA1 P30542 1/20 0.42
CDK1 P06493 1/20 0.41
CDK5 Q00535 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL292922 1.00 ADORA2A (0.54) ADORA2AADORA3CCNE2CCNA2CCNE1
Trifluoroacetic Acid SCHEMBL242659 0.96 ADORA2A (0.51) ADORA2AADORA3CCNE2CCNA2CCNE1
SCHEMBL242569 0.94 ADORA2A (0.55) ADORA2AADORA3CCNE2CCNA2CCNE1
SCHEMBL242568 0.94 ADORA2A (0.55) ADORA2AADORA3CCNE2CCNA2CCNE1
SCHEMBL1401995 0.94 ADORA2A (0.60) ADORA2AADORA3CCNE2CCNA2CCNE1
SCHEMBL1401992 0.94 ADORA2A (0.60) ADORA2AADORA3CCNE2CCNA2CCNE1
Hydrochloric Acid SCHEMBL241391 0.94 ADORA2A (0.47) ADORA2AADORA3CCNE2CCNA2CCNE1
Hydrochloric Acid SCHEMBL241392 0.94 ADORA2A (0.47) ADORA2AADORA3CCNE2CCNA2CCNE1
SCHEMBL239194 0.94 ADORA2A (0.62) ADORA2AADORA3CCNE2CCNA2CCNE1
SCHEMBL13879042 0.94 ADORA2A (0.62) ADORA2AADORA3CCNE2CCNA2CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013211-B1 PURINE DERIVATIVES FOR USE AS ADENOSIN A2A RECEPTOR AGONISTS NOVARTIS AG (CH) 2012-03-14 EP disclosed