SCHEMBL2930703

SCHEMBL2930703

CC(C)Oc1c2c(c(OC(C)C)c3ccccc13)C(=O)N(c1ccc(CC=O)cc1Br)C2=O

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 4/20 0.39
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA7 P43166 2/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
GRM4 Q14833 1/20 0.32
TP53 P04637 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2930584 0.85 PTGER4 (0.52) PTGER4CYP1A2CYP2D6
SCHEMBL2926785 0.85 PTGER4 (0.55) PTGER4CYP1A2CYP2D6
SCHEMBL10079622 0.83 PTGER4 (0.37) PTGER4CYP1A2CYP2D6
SCHEMBL13177685 0.81 PTGER4 (0.47) PTGER4CYP1A2CYP2D6
SCHEMBL10078896 0.80 PTGER4 (0.40) PTGER4CYP1A2CYP2D6
SCHEMBL13594947 0.78 PTGER4 (0.47) PTGER4CYP1A2CYP2D6
SCHEMBL10078418 0.76 PTGER4 (0.37) PTGER4CYP1A2CYP2D6CA1CA2
SCHEMBL10078916 0.76 PTGER4 (0.46) PTGER4CYP1A2CYP2D6
SCHEMBL13594923 0.76 PTGER4 (0.48) PTGER4CYP1A2CYP2D6MAPT
SCHEMBL13594930 0.75 PTGER4 (0.48) PTGER4CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081897-B1 ISOINDOL DERIVATIVES AS EP4 RECEPTOR AGONISTS GLAXO GROUP LTD (GB) 2010-09-15 EP disclosed