SCHEMBL2931846

SCHEMBL2931846

Cc1ncc(C#N)c(Nc2ccc3[nH]ccc3c2C)c1C=Cc1ccc(CO)cn1

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PRKCQ Q04759 20/20 0.60
PRKCD Q05655 20/20 0.60
PRKCH P24723 1/20 0.54
PRKCE Q02156 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13820173 1.00 PRKCQ (0.60) PRKCQPRKCDPRKCHPRKCE
SCHEMBL2927042 0.88 PRKCQ (0.76) PRKCQPRKCD
SCHEMBL2927039 0.88 PRKCQ (0.76) PRKCQPRKCD
SCHEMBL2928637 0.85 PRKCQ (0.60) PRKCQPRKCDPRKCHPRKCE
SCHEMBL2929219 0.85 PRKCQ (0.81) PRKCQPRKCDPRKCHPRKCE
SCHEMBL2929221 0.85 PRKCQ (0.81) PRKCQPRKCDPRKCHPRKCE
SCHEMBL2980036 0.85 PRKCQ (0.69) PRKCQPRKCD
SCHEMBL2932024 0.84 PRKCQ (0.61) PRKCQPRKCDPRKCHPRKCE
SCHEMBL2932023 0.84 PRKCQ (0.61) PRKCQPRKCDPRKCHPRKCE
SCHEMBL2934644 0.83 PRKCQ (0.76) PRKCQPRKCDPRKCHPRKCE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229377-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS Wyeth LLC (US) 2010-09-22 EP disclosed
WO-2009076602-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS WYETH (US) 2009-06-18 WO disclosed