SCHEMBL29329889

SCHEMBL29329889

COCc1nc(O)c2c(n1)CN(C(=O)OC(C)(C)C)CC2

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.44
TNKS2 Q9H2K2 1/20 0.44
PARP2 Q9UGN5 1/20 0.44
ESR2 Q92731 1/20 0.44
ADORA1 P30542 2/20 0.41
MTOR P42345 2/20 0.40
MAPT P10636 3/20 0.39
NR1H2 P55055 1/20 0.38
KDM4E B2RXH2 1/20 0.38
P2RX3 P56373 7/20 0.37
F12 P00748 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29329891 0.87 PARP1 (0.43) PARP1TNKS2PARP2ESR2ADORA1
SCHEMBL29330189 0.82 PARP1 (0.46) PARP1TNKS2PARP2ESR2ADORA1
SCHEMBL13250465 0.82 PARP1 (0.47) PARP1TNKS2PARP2ESR2ADORA1
SCHEMBL30776241 0.82 PARP1 (0.47) PARP1TNKS2PARP2ESR2ADORA1
SCHEMBL3264705 0.81 ADORA1 (0.49) PARP1TNKS2PARP2ESR2ADORA1
SCHEMBL22720588 0.80 PARP1 (0.47) PARP1TNKS2PARP2ESR2ADORA1
SCHEMBL19616687 0.79 PARP1 (0.45) PARP1TNKS2PARP2ESR2ADORA1
SCHEMBL16034353 0.79 PARP1 (0.45) PARP1TNKS2PARP2ESR2ADORA1
SCHEMBL9951661 0.79 PARP1 (0.45) PARP1TNKS2PARP2ESR2ADORA1
SCHEMBL29330064 0.78 PARP1 (0.43) PARP1TNKS2PARP2ESR2ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4400500-A1 HALOGEN-SUBSTITUTED PYRIDAZINONE COMPOUND AND APPLICATION THEREOF Medshine Discovery Inc. (CN) 2024-07-17 EP disclosed