SCHEMBL29330190

SCHEMBL29330190

COc1nc(Cl)c2c(n1)CN(C(=O)OC(C)(C)C)CC2

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.45
TNKS2 Q9H2K2 1/20 0.45
PARP2 Q9UGN5 1/20 0.45
ADORA1 P30542 2/20 0.45
ESR2 Q92731 1/20 0.43
MAPT P10636 3/20 0.41
KDM4E B2RXH2 1/20 0.41
NR1H2 P55055 1/20 0.39
MTOR P42345 1/20 0.39
MKNK1 Q9BUB5 2/20 0.39
POLB P06746 1/20 0.38
P2RX3 P56373 5/20 0.38
F12 P00748 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29330189 0.86 PARP1 (0.46) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL1832511 0.86 PARP1 (0.47) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL16033863 0.85 PARP1 (0.47) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL31246480 0.84 PARP1 (0.43) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL16034060 0.83 PARP1 (0.45) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL29329891 0.82 PARP1 (0.43) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL24730853 0.82 PARP1 (0.45) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL10166308 0.82 PARP1 (0.45) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL29899536 0.82 PARP1 (0.47) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL29330065 0.81 PARP1 (0.43) PARP1TNKS2PARP2ADORA1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4400500-A1 HALOGEN-SUBSTITUTED PYRIDAZINONE COMPOUND AND APPLICATION THEREOF Medshine Discovery Inc. (CN) 2024-07-17 EP disclosed