SCHEMBL2933209

SCHEMBL2933209

Cc1c(Nc2c(C#N)cncc2C=CCN2CCCCC2)ccc2[nH]ccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCQ Q04759 20/20 1.00
PRKCD Q05655 20/20 1.00
LYN P07948 3/20 0.85
PRKCH P24723 3/20 0.85
PRKCE Q02156 3/20 0.85
LCK P06239 2/20 0.72
PRKCB P05771 1/20 0.72
CHEK1 O14757 1/20 0.71
IKBKB O14920 1/20 0.71
CHUK O15111 1/20 0.71
ABL1 P00519 1/20 0.71
FYN P06241 1/20 0.71
CDK1 P06493 1/20 0.71
MET P08581 1/20 0.71
HCK P08631 1/20 0.71
SRC P12931 1/20 0.71
PDGFRA P16234 1/20 0.71
CDK2 P24941 1/20 0.71
AKT1 P31749 1/20 0.71
KDR P35968 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2933205 1.00 PRKCQ (1.00) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2928798 0.99 PRKCQ (0.98) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2928799 0.99 PRKCQ (0.98) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2932107 0.92 PRKCQ (1.00) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2932101 0.92 PRKCQ (1.00) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2927191 0.92 PRKCQ (1.00) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2927188 0.92 PRKCQ (1.00) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2935862 0.91 PRKCQ (1.00) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2935865 0.91 PRKCQ (1.00) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2935807 0.91 PRKCQ (1.00) PRKCQPRKCDLYNPRKCHPRKCE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229377-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS Wyeth LLC (US) 2010-09-22 EP claimed
WO-2009076602-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS WYETH (US) 2009-06-18 WO claimed