SCHEMBL2934737

SCHEMBL2934737

NC(=O)Nc1sc(-c2ccc(OC3CCCC3)cc2OCCN2CCCCC2)cc1OC(N)=O

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 3/20 0.51
MET P08581 1/20 0.43
KDM4E B2RXH2 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KMT2A Q03164 1/20 0.36
HRH3 Q9Y5N1 2/20 0.35
ESR1 P03372 2/20 0.35
ESR2 Q92731 2/20 0.35
PSMB1 P20618 1/20 0.35
PSMB5 P28074 1/20 0.35
PSMB2 P49721 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1929738 0.89 CHEK1 (0.65) CHEK1METKDM4EKMT2A
SCHEMBL2934974 0.86 CHEK1 (0.54) CHEK1METKDM4ESMN1; SMN2HRH3
SCHEMBL2935301 0.85 CHEK1 (0.52) CHEK1KDM4ESMN1; SMN2KMT2AHRH3
SCHEMBL2932598 0.85 CHEK1 (0.52) CHEK1KDM4ESMN1; SMN2KMT2AHRH3
SCHEMBL2932580 0.81 CHEK1 (0.47) CHEK1KDM4EKMT2AHRH3
SCHEMBL2933542 0.80 CHEK1 (0.46) CHEK1KMT2AHRH3
SCHEMBL1928162 0.75 CHEK1 (0.69) CHEK1METKDM4EKMT2A
SCHEMBL1930902 0.74 CHEK1 (0.67) CHEK1KDM4EKMT2A
SCHEMBL1927323 0.74 CHEK1 (0.67) CHEK1KDM4EKMT2A
SCHEMBL1928564 0.70 CHEK1 (0.61) CHEK1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1421074-B1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2010-09-29 EP claimed