SCHEMBL2935875

SCHEMBL2935875

Cc1c(Nc2c(C#N)cncc2/C=C/CCN2CCOCC2)ccc2[nH]ccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PRKCQ Q04759 20/20 1.00
PRKCD Q05655 20/20 1.00
PRKCB P05771 2/20 0.83
LCK P06239 2/20 0.83
LYN P07948 2/20 0.83
PRKCH P24723 2/20 0.83
PRKCE Q02156 2/20 0.83

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2935878 1.00 PRKCQ (1.00) PRKCQPRKCDPRKCBLCKLYN
SCHEMBL2931489 0.95 PRKCQ (1.00) PRKCQPRKCDPRKCBLCKLYN
SCHEMBL2931484 0.95 PRKCQ (1.00) PRKCQPRKCDPRKCBLCKLYN
SCHEMBL2983372 0.93 PRKCQ (0.98) PRKCQPRKCDPRKCBLCKLYN
SCHEMBL2935862 0.92 PRKCQ (1.00) PRKCQPRKCDPRKCBLCKLYN
SCHEMBL2935804 0.92 PRKCQ (1.00) PRKCQPRKCDPRKCBLCKLYN
SCHEMBL2935865 0.92 PRKCQ (1.00) PRKCQPRKCDPRKCBLCKLYN
SCHEMBL2935807 0.92 PRKCQ (1.00) PRKCQPRKCDPRKCBLCKLYN
SCHEMBL2928581 0.91 PRKCQ (1.00) PRKCQPRKCDPRKCBLCKLYN
SCHEMBL2928579 0.91 PRKCQ (1.00) PRKCQPRKCDPRKCBLCKLYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229377-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS Wyeth LLC (US) 2010-09-22 EP disclosed
WO-2009076602-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS WYETH (US) 2009-06-18 WO disclosed