SCHEMBL29360565

SCHEMBL29360565

O=C(NC1CCCc2ccccc21)c1cc(C2CCN(C(=O)Cn3nc(C(F)F)cc3C3CC3)CC2)ccn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.41
ALDH1A1 P00352 9/20 0.40
KDM4E B2RXH2 5/20 0.40
HPGD P15428 5/20 0.40
KMT2A Q03164 3/20 0.39
LMNA P02545 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MAPT P10636 1/20 0.39
CYP2D6 P10635 3/20 0.39
TAS1R3 Q7RTX0 2/20 0.39
TAS1R1 Q7RTX1 2/20 0.39
TAS1R2 Q8TE23 2/20 0.39
MEN1 O00255 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C19 P33261 2/20 0.39
HTT P42858 2/20 0.38
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
CYP1A2 P05177 2/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18112867 1.00 TSHR (0.41) TSHRALDH1A1KDM4EHPGDKMT2A
SCHEMBL19176075 1.00 TSHR (0.41) TSHRALDH1A1KDM4EHPGDKMT2A
SCHEMBL29360345 0.92 TSHR (0.42) TSHRALDH1A1KDM4EHPGDKMT2A
SCHEMBL19176162 0.92 TSHR (0.42) TSHRALDH1A1KDM4EHPGDKMT2A
SCHEMBL18112863 0.92 TSHR (0.42) TSHRALDH1A1KDM4EHPGDKMT2A
SCHEMBL29538537 0.91 TSHR (0.42) TSHRALDH1A1KDM4EHPGDKMT2A
SCHEMBL19176174 0.91 TSHR (0.45) TSHRALDH1A1KDM4EHPGDKMT2A
SCHEMBL18112859 0.91 TSHR (0.45) TSHRALDH1A1KDM4EHPGDKMT2A
SCHEMBL29362208 0.91 TSHR (0.45) TSHRALDH1A1KDM4EHPGDKMT2A
SCHEMBL18112862 0.91 TSHR (0.41) TSHRALDH1A1KDM4EHPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 105 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4710766-A1 MIXTURES OF AMBRUTICIN WITH AT LEAST ONE FURTHER PESTICIDE BASF SE (DE) 2026-03-18 EP claimed
WO-2025223904-A1 MIXTURES OF STROBILURIN TYPE COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI CONTAINING AN AMINO ACID SUBSTITUTION F129L IN THE MITOCHONDRIAL CYTOCHROME B PROTEIN CONFERRING RESISTANCE TO QO INHIBITORS WITH AT LEAST ONE FURTHER PESTICIDE I BASF SE (DE) 2025-10-30 WO claimed
EP-4618761-A1 FUNGICIDAL MIXTURE COMPRISING SUBSTITUTED PYRIDINES BASF SE (DE) 2025-09-24 EP claimed
EP-4618760-A1 FUNGICIDAL MIXTURE COMPRISING SUBSTITUTED PYRIDINES BASF SE (DE) 2025-09-24 EP claimed
WO-2024104814-A1 FUNGICIDAL MIXTURE COMPRISING SUBSTITUTED PYRIDINES BASF SE (DE) 2024-05-23 WO claimed
EP-4346412-A1 FUNGICIDAL COMPOSITION CONTAINING OXADIAZOLE COMPOUNDS PI Industries Ltd. (IN) 2024-04-10 EP claimed
CN-117396074-A Fungicidal compositions containing oxadiazole compounds PI工业有限公司 2024-01-12 CN claimed
CN-116634876-A Mixtures and compositions comprising Fusarium A, fusarium B and fungicides 巴斯夫欧洲公司 2023-08-22 CN claimed
WO-2022249074-A1 FUNGICIDAL COMPOSITION CONTAINING OXADIAZOLE COMPOUNDS PI INDUSTRIES LTD. (IN) 2022-12-01 WO claimed
WO-2022136003-A1 MIXTURES AND COMPOSITIONS COMPRISING FUSARICIDIN A, FUSARICIDIN B AND FUNGICIDES BASF SE (DE) 2022-06-30 WO claimed
EP-4739690-A1 SUBSTITUTED QUINOLYL/QUINOXALYL DIHYDROPYRROLOTRIAZINE COMPOUNDS FOR COMBATTING PHYTO-PATHOGENIC FUNGI BASF SE (DE) 2026-05-13 EP disclosed
EP-4739691-A1 SUBSTITUTED PYRIDYL/PYRAZINYL DIHYDROPYRROLOTRIAZINE COMPOUNDS FOR COMBATTING PHYTOPATH-OGENIC FUNGI BASF SE (DE) 2026-05-13 EP disclosed
EP-4702006-A1 USE OF STROBILURIN TYPE COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI CONTAINING AN AMINO ACID SUBSTITUTION F129L IN THE MITOCHONDRIAL CYTOCHROME B PROTEIN CONFERRING RESISTANCE TO QO INHIBITORS XVI BASF SE (DE) 2026-03-04 EP disclosed
EP-4680605-A1 SUBSTITUTED PYRIDYL/PYRAZIDYL DIHYDROBENZOTHIAZEPINE COMPOUNDS FOR COMBATTING PHYTOPATHOGENIC FUNGI BASF SE (DE) 2026-01-21 EP disclosed
EP-4662210-A1 NEW SUBSTITUTED QUINOLINE COMPOUNDS FOR COMBATITNG PHYTOPATHOGENIC FUNGI BASF SE (DE) 2025-12-17 EP disclosed
WO-2022090071-A1 USE OF MEFENPYR-DIETHYL FOR CONTROLLING PHYTOPATHOGENIC FUNGI BASF SE (DE) 2022-05-05 WO disclosed
EP-3975718-A1 MESOIONIC IMIDAZOLIUM COMPOUNDS AND DERIVATIVES FOR COMBATING ANIMAL PESTS BASF SE (DE) 2022-04-06 EP disclosed
CN-114174267-A Pesticidal pyrazole and triazole derivatives 巴斯夫欧洲公司 2022-03-11 CN disclosed
WO-2022033906-A1 USE OF STROBILURIN TYPE COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI CONTAINING AN AMINO ACID SUBSTITUTION F129L IN THE MITOCHONDRIAL CYTOCHROME B PROTEIN CONFERRING RESISTANCE TO QO INHIBITORS VIII BASF SE (DE) 2022-02-17 WO disclosed
WO-2022017836-A1 FUNGICIDAL COMPOSITIONS COMPRISING (R)-2-[4-(4-CHLOROPHENOXY)-2-(TRIFLUOROMETHYL)PHENYL]-1- (1,2,4-TRIAZOL-1-YL)PROPAN-2-OL BASF Agro B.V. (NL) 2022-01-27 WO disclosed