Azd2461

Azd2461

SCHEMBL29361302

COC1CCN(C(=O)c2cc(Cc3n[nH]c(=O)c4ccccc34)ccc2F)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 20/20 1.00
PRAP1 Q96NZ9 1/20 1.00
TNKS O95271 1/20 0.75
ADORA1 P30542 1/20 0.75
CDK6 Q00534 1/20 0.75
PDE3A Q14432 1/20 0.75
PARP6 Q2NL67 1/20 0.75
PARP15 Q460N3 1/20 0.75
PARP14 Q460N5 1/20 0.75
PARP10 Q53GL7 1/20 0.75
TIPARP Q7Z3E1 1/20 0.75
PARP8 Q8N3A8 1/20 0.75
PARP16 Q8N5Y8 1/20 0.75
PARP12 Q9H0J9 1/20 0.75
TNKS2 Q9H2K2 1/20 0.75
PARP11 Q9NR21 1/20 0.75
PARP2 Q9UGN5 1/20 0.75
PARP4 Q9UKK3 1/20 0.75
PARP3 Q9Y6F1 1/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Azd2461 SCHEMBL77012 1.00 PARP1 (1.00) PARP1PRAP1TNKSADORA1CDK6
Azd2461 SCHEMBL29360368 1.00 PARP1 (1.00) PARP1PRAP1TNKSADORA1CDK6
SCHEMBL22852674 0.97 PARP1 (1.00) PARP1PRAP1TNKSADORA1CDK6
SCHEMBL22852672 0.95 PARP1 (1.00) PARP1PRAP1TNKSADORA1CDK6
SCHEMBL31311843 0.92 PARP1 (0.85) PARP1PRAP1TNKSADORA1CDK6
SCHEMBL76871 0.91 PARP1 (0.84) PARP1PRAP1TNKSADORA1CDK6
SCHEMBL87500 0.91 PARP1 (0.84) PARP1PRAP1TNKSADORA1CDK6
SCHEMBL22852677 0.91 PARP1 (1.00) PARP1PRAP1TNKSADORA1CDK6
SCHEMBL78156 0.91 PARP1 (0.83) PARP1PRAP1TNKSADORA1CDK6
SCHEMBL86912 0.91 PARP1 (0.82) PARP1PRAP1TNKSADORA1CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 231 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026106998-A1 PROSTATE-SPECIFIC MEMBRANE ANTIGEN (PSMA)-TARGETED POLY(ADP-RIBOSE) POLYMERASE (PARP) INHIBITOR AND RELATED COMPOSITION AND METHOD OF USE PURDUE RESEARCH FOUNDATION (US) 2026-05-21 WO claimed
EP-4739310-A1 ECTONUCLEOTIDE PYROPHOSPHATASE/PHOSPHODIESTERASE 1 (ENPP1) INHIBITOR COMBINATIONS AND USES THEREOF Insilico Medicine IP Limited (HK) 2026-05-13 EP claimed
US-20250223292-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED 2025-07-10 US claimed
US-20250100977-A1 MERCAPTOPYRIMIDINE COMPOUNDS THAT INHIBIT NONHOMOLOGOUS END JOINING AND METHODS THEREOF UNIVERSITY OF MYSORE (IN) 2025-03-27 US claimed
EP-4190786-B1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMA (US) 2025-02-26 EP claimed
WO-2025007955-A1 ECTONUCLEOTIDE PYROPHOSPHATASE/PHOSPHODIESTERASE 1 (ENPP1) INHIBITOR COMBINATIONS AND USES THEREOF INSILICO MEDICINE IP LIMITED (CN) 2025-01-09 WO claimed
EP-4479046-A2 METHODS TO PREVENT THERAPY RESISTANCE IN MELANOMA VIA BLOCKING GENOMIC INSTABILITY The Regents of University of California (US) 2024-12-25 EP claimed
WO-2024217502-A1 METHIONINE ADENOSYLTRANSFERASE 2A (MAT2A) INHIBITOR COMBINATIONS AND USES THEREOF INSILICO MEDICINE IP LIMITED (CN) 2024-10-24 WO claimed
WO-2024216115-A1 METHODS FOR PRODUCING A SUPER CENTRAL MEMORY CD8 T CELL SUBTYPE BY POLY(ADP-RIBOSE) POLYMERASE (PARP) INHIBITION AND USES THEREOF GEORGETOWN UNIVERSITY (US) 2024-10-17 WO claimed
WO-2024186926-A1 STRATEGIES TO PREVENT THE EVOLUTION OF LETHAL, MULTI-THERAPY-RESISTANT, WIDELY METASTATIC CUTANEOUS MELANOMA THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-09-12 WO claimed
EP-4294844-A1 COMBINATION THERAPIES WITH ANTI-CD38 ANTIBODIES AND PARP OR ADENOSINE RECEPTOR INHIBITORS Janssen Biotech, Inc. (US) 2023-12-27 EP claimed
WO-2023158911-A2 METHODS TO PREVENT THERAPY RESISTANCE IN MELANOMA VIA BLOCKING GENOMIC INSTABILITY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-08-24 WO claimed
WO-2023126980-A1 MERCAPTOPYRIMIDINE COMPOUNDS THAT INHIBIT NONHOMOLOGOUS END JOINING AND METHODS THEREOF INDIAN INSTITUTE OF SCIENCE (IN) 2023-07-06 WO claimed
EP-4190786-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE Vertex Pharmaceuticals Incorporated (US) 2023-06-07 EP claimed
US-20230123585-A1 COMPOSITIONS AND METHODS FOR TREATING OR PREVENTING CANCER USING DEUBIQUITINASE INHIBITORS UNIV CHICAGO (US) 2023-04-20 US claimed
EP-3808749-B1 PYRAZOLO[1,5-A]PYRIMIDINES USEFUL AS INHIBITORS OF ATR KINASE FOR THE TREATMENT OF CANCER DISEASES VERTEX PHARMA (US) 2023-03-08 EP claimed
EP-4065097-A1 PARTHANATOS CELL DEATH INHIBITORS FOR USE IN THE TREATMENT OF PSORIASIS Universidad De Murcia (ES) 2022-10-05 EP claimed
US-20220275090-A1 Combination Therapies with Anti-CD38 Antibodies and PARP or Adenosine Receptor Inhibitors JANSSEN BIOTECH, INC. 2022-09-01 US claimed
WO-2022175920-A1 COMBINATION THERAPIES WITH ANTI-CD38 ANTIBODIES AND PARP OR ADENOSINE RECEPTOR INHIBITORS JANSSEN BIOTECH, INC. (US) 2022-08-25 WO claimed
US-20220233521-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE AND COMBINATION THERAPIES THEREOF VERTEX PHARMACEUTICALS INCORPORATED 2022-07-28 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220275090-A1 Combination Therapies with Anti-CD38 Antibodies and PARP or Adenosine Receptor Inhibitors CD38, PARP1, PARP11 PARP1 2/4885PRAP1 467/4885TNKS 47/4885
US-20250100977-A1 MERCAPTOPYRIMIDINE COMPOUNDS THAT INHIBIT NONHOMOLOGOUS END JOINING AND METHODS THEREOF LIG4, LIG1, LIG3 PARP1 39/4885PRAP1 1737/4885TNKS 120/4885
US-20250223292-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE ATR, MAP3K20, CHEK1 PARP1 339/4885PRAP1 2202/4885TNKS 44/4885
US-20220233521-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE AND COMBINATION THERAPIES THEREOF ATR, CHEK1, CHEK2 PARP1 159/4885PRAP1 1889/4885TNKS 31/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.