SCHEMBL2937062

SCHEMBL2937062

CN(C)C(=O)C(=O)N(C)C1CCCCn2c1nc(C(=O)NCc1ccc(F)cc1)c(O)c2=O.COC(=O)C(=O)Cl

nearest known ligand 0.87

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.87
KCNH2 Q12809 1/20 0.63
CALCA P06881 3/20 0.39
KCNE1 P15382 1/20 0.39
CCR1 P32246 1/20 0.39
KCNQ1 P51787 1/20 0.39
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.35
ERCC1 P07992 1/20 0.35
FEN1 P39748 1/20 0.35
ERCC4 Q92889 1/20 0.35
LIPG Q9Y5X9 1/20 0.34
POLB P06746 2/20 0.34
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL420510 0.93 CYP2C9 (1.00) CYP2C9KCNH2CALCAKCNE1CCR1
SCHEMBL1749374 0.91 CYP2C9 (0.95) CYP2C9KCNH2CALCAKCNE1CCR1
SCHEMBL1376381 0.85 CYP2C9 (0.81) CYP2C9KCNH2CALCAKCNE1CCR1
SCHEMBL13419820 0.85 CYP2C9 (0.83) CYP2C9KCNH2CALCAKCNE1CCR1
SCHEMBL1376921 0.84 CYP2C9 (0.80) CYP2C9KCNH2MAPTSMN1; SMN2MEN1
SCHEMBL12529638 0.84 CYP2C9 (0.77) CYP2C9KCNH2CALCAKCNE1CCR1
SCHEMBL1378080 0.84 CYP2C9 (0.77) CYP2C9KCNH2CALCAMAPTSMN1; SMN2
SCHEMBL1749433 0.84 CYP2C9 (0.79) CYP2C9KCNH2CALCAMAPTMEN1
SCHEMBL1378474 0.83 CYP2C9 (0.81) CYP2C9KCNH2CALCAKCNE1CCR1
SCHEMBL1379153 0.83 CYP2C9 (0.76) CYP2C9KCNH2CALCAMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1578748-B1 TETRAHYDRO-4H-PYRIDO[1,2-A]PYRIMIDINES AND RELATED COMPOUNDS USEFUL AS HIV INTEGRASE INHIBITORS ANGELETTI P IST RICHERCHE BIO (IT) 2010-09-15 EP disclosed