SCHEMBL29370855

SCHEMBL29370855

CN1CCN(c2cccc(Nc3ncc4cccc(-c5ccc(N6CCOCC6)cc5)c4n3)c2)CC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTK P33981 1/20 0.61
JAK2 O60674 6/20 0.61
BRD4 O60885 2/20 0.61
MAPK10 P53779 5/20 0.56
JUN P05412 4/20 0.56
MAPK8 P45983 4/20 0.56
FGFR1 P11362 1/20 0.53
KDR P35968 1/20 0.53
CCNT1 O60563 1/20 0.52
CCNE1 P24864 1/20 0.52
CDK2 P24941 1/20 0.52
CDK9 P50750 1/20 0.52
JAK3 P52333 3/20 0.51
PTK2 Q05397 3/20 0.51
JAK1 P23458 1/20 0.51
RIPK2 O43353 2/20 0.50
HDAC3 O15379 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18376727 1.00 TTK (0.61) TTKJAK2BRD4MAPK10JUN
SCHEMBL18376233 0.94 JAK2 (0.63) TTKJAK2BRD4MAPK10JUN
SCHEMBL18377031 0.92 JAK2 (0.55) TTKJAK2BRD4MAPK10JUN
SCHEMBL18376225 0.89 JAK2 (0.59) TTKJAK2BRD4FGFR1KDR
SCHEMBL18376589 0.89 JAK2 (0.58) TTKJAK2BRD4FGFR1KDR
SCHEMBL29371805 0.89 JAK2 (0.58) TTKJAK2BRD4FGFR1KDR
SCHEMBL29371867 0.89 JAK2 (0.60) JAK2BRD4FGFR1KDRCCNT1
SCHEMBL18376722 0.89 JAK2 (0.60) JAK2BRD4FGFR1KDRCCNT1
SCHEMBL30859695 0.88 TTK (0.65) TTKJAK2MAPK10JUNMAPK8
SCHEMBL18376252 0.88 TTK (0.65) TTKJAK2MAPK10JUNMAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113999180-A Quinazoline compound, intermediate thereof, preparation method, pharmaceutical composition and application 上海医药集团股份有限公司 2022-02-01 CN claimed
CN-113999180-B Quinazoline compound, intermediate, preparation method, pharmaceutical composition and application 上海医药集团股份有限公司 2024-03-26 CN disclosed
CN-113999180-A Quinazoline compound, intermediate thereof, preparation method, pharmaceutical composition and application 上海医药集团股份有限公司 2022-02-01 CN disclosed