SCHEMBL29388366

SCHEMBL29388366

CCn1cnc2c(N)nc(SC)nc21

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 2/20 0.67
CCNB1 P14635 2/20 0.67
CCNE1 P24864 2/20 0.67
CDK2 P24941 2/20 0.67
ADORA2A P29274 5/20 0.55
ADORA1 P30542 4/20 0.55
PI4KA P42356 1/20 0.55
PI4K2B Q8TCG2 1/20 0.55
PI4K2A Q9BTU6 1/20 0.55
PI4KB Q9UBF8 1/20 0.55
ADORA2B P29275 2/20 0.48
TMIGD3 P0DMS9 2/20 0.48
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
P2RY1 P47900 2/20 0.40
ENPP1 P22413 2/20 0.39
P2RY12 Q9H244 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29388387 0.86 CDK1 (0.65) CDK1CCNB1CCNE1CDK2ADORA2A
SCHEMBL24701698 0.84 CDK1 (0.61) CDK1CCNB1CCNE1CDK2ADORA2A
SCHEMBL21282838 0.81 CDK1 (0.46) CDK1CCNB1CCNE1CDK2ADORA2A
SCHEMBL19503597 0.81 CDK1 (0.45) CDK1CCNB1CCNE1CDK2ADORA2A
SCHEMBL19503305 0.81 CDK1 (0.45) CDK1CCNB1CCNE1CDK2ADORA2A
SCHEMBL19553855 0.80 ADORA2A (0.53) CDK1CCNB1CCNE1CDK2ADORA2A
SCHEMBL7205020 0.80 PDE4A (0.62) CDK1ADORA2AADORA1PI4KAPI4K2B
SCHEMBL8767031 0.80 CCNE1 (1.00) CDK1CCNB1CCNE1CDK2ADORA2A
SCHEMBL14619182 0.79 CDK1 (0.60) CDK1CCNB1CCNE1CDK2ADORA2A
SCHEMBL5161756 0.79 CDK1 (0.73) CDK1CCNB1CCNE1CDK2ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3955929-A1 NEW PYRIMIDINE DERIVATIVES FOR PREVENTION AND TREATMENT OF GRAM-NEGATIVE BACTERIAL INFECTION, CONTAMINATION AND FOULING Université de Liège (BE) 2022-02-23 EP claimed
EP-3955929-A1 NEW PYRIMIDINE DERIVATIVES FOR PREVENTION AND TREATMENT OF GRAM-NEGATIVE BACTERIAL INFECTION, CONTAMINATION AND FOULING Université de Liège (BE) 2022-02-23 EP disclosed