SCHEMBL29401291

SCHEMBL29401291

CCn1c(CO)nn(-c2ccc3c(=O)n(-c4cccc(F)c4)nc(C(C)C)c3c2)c1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 20/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22552377 1.00 DHODH (1.00) DHODH
SCHEMBL29401296 0.87 DHODH (1.00) DHODH
SCHEMBL22552252 0.87 DHODH (1.00) DHODH
SCHEMBL29480969 0.85 DHODH (0.75) DHODH
SCHEMBL22552147 0.85 DHODH (1.00) DHODH
SCHEMBL29404137 0.85 DHODH (1.00) DHODH
SCHEMBL22552199 0.85 DHODH (1.00) DHODH
SCHEMBL29403725 0.85 DHODH (1.00) DHODH
SCHEMBL22552241 0.83 DHODH (1.00) DHODH
SCHEMBL29403542 0.83 DHODH (1.00) DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114174278-B Dihydroorotate dehydrogenase inhibitors 詹森生物科技公司 2024-08-23 CN claimed
WO-2022074534-A1 COMBINATIONS OF DIHYDROOROTATE DEHYDROGENASE INHIBITORS AND HYPOMETHYLATING AGENTS JANSSEN BIOTECH, INC. (US) 2022-04-14 WO claimed
CN-114174278-A Dihydroorotate dehydrogenase inhibitors 詹森生物科技公司 2022-03-11 CN claimed
EP-3956320-A1 DIHYDROOROTATE DEHYDROGENASE INHIBITORS Janssen Biotech, Inc. (US) 2022-02-23 EP claimed
EP-4626427-A1 COMBINATIONS COMPRISING A MENIN-MLL INHIBITOR AND A BCL-2 INHIBITOR Janssen Pharmaceutica NV (BE) 2025-10-08 EP disclosed
EP-4626426-A1 COMBINATIONS COMPRISING A MENIN-MLL INHIBITOR AND AT LEAST ONE OTHER THERAPEUTIC AGENT JANSSEN Pharmaceutica NV (BE) 2025-10-08 EP disclosed
CN-118845786-A Combination therapy 詹森药业有限公司 2024-10-29 CN disclosed
CN-118845787-A Combination therapy 詹森药业有限公司 2024-10-29 CN disclosed
CN-114174278-B Dihydroorotate dehydrogenase inhibitors 詹森生物科技公司 2024-08-23 CN disclosed
WO-2024114666-A1 COMBINATIONS COMPRISING A MENIN-MLL INHIBITOR AND A BCL-2 INHIBITOR JANSSEN PHARMACEUTICA NV (BE) 2024-06-06 WO disclosed
WO-2024114664-A1 COMBINATIONS COMPRISING A MENIN-MLL INHIBITOR AND AT LEAST ONE OTHER THERAPEUTIC AGENT JANSSEN PHARMACEUTICA NV (BE) 2024-06-06 WO disclosed
EP-4337215-A1 COMBINATION THERAPIES JANSSEN Pharmaceutica NV (BE) 2024-03-20 EP disclosed
CN-117460513-A Combination therapy 詹森药业有限公司 2024-01-26 CN disclosed
WO-2022237719-A1 COMBINATION THERAPIES JANSSEN PHARMACEUTICA NV (BE) 2022-11-17 WO disclosed
WO-2022237720-A1 COMBINATION THERAPIES JANSSEN PHARMACEUTICA NV (BE) 2022-11-17 WO disclosed
WO-2022074534-A1 COMBINATIONS OF DIHYDROOROTATE DEHYDROGENASE INHIBITORS AND HYPOMETHYLATING AGENTS JANSSEN BIOTECH, INC. (US) 2022-04-14 WO disclosed
CN-114174278-A Dihydroorotate dehydrogenase inhibitors 詹森生物科技公司 2022-03-11 CN disclosed
EP-3956320-A1 DIHYDROOROTATE DEHYDROGENASE INHIBITORS Janssen Biotech, Inc. (US) 2022-02-23 EP disclosed