Prothioconazole-Desthio

Prothioconazole-Desthio

SCHEMBL29405397

OC(Cc1ccccc1Cl)(Cn1cncn1)C1(Cl)CC1

nearest known ligand 0.45

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.45
KMT2A Q03164 1/20 0.39
CYP3A4 P08684 2/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP19A1 P11511 3/20 0.38
CACNA1G O43497 1/20 0.36
CACNA1H O95180 1/20 0.36
CACNA1I Q9P0X4 1/20 0.36
FDPS P14324 1/20 0.35
LMNA P02545 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
CYP2C19 P33261 1/20 0.35
ADRA1A P35348 1/20 0.35
CYP51A1 Q16850 1/20 0.35
KDM4E B2RXH2 1/20 0.35
PDCD1 Q15116 2/20 0.34
CD274 Q9NZQ7 2/20 0.34
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Prothioconazole-Desthio SCHEMBL2491761 1.00 HSP90AA1 (0.45) HSP90AA1KMT2ACYP3A4ALDH1A1CYP19A1
Prothioconazole-Desthio SCHEMBL8975106 0.92 CYP3A4 (0.47) HSP90AA1KMT2ACYP3A4ALDH1A1CYP19A1
SCHEMBL8937971 0.87 HSP90AA1 (0.44) HSP90AA1KMT2ACYP3A4ALDH1A1CYP19A1
SCHEMBL16165981 0.86 KMT2A (0.38) HSP90AA1KMT2ACYP3A4ALDH1A1CYP19A1
SCHEMBL10385481 0.86 KMT2A (0.43) HSP90AA1KMT2ACYP3A4ALDH1A1CYP19A1
SCHEMBL28701737 0.85 HSP90AA1 (0.42) HSP90AA1KMT2ACYP3A4ALDH1A1CYP19A1
SCHEMBL9682964 0.85 HSP90AA1 (0.42) HSP90AA1KMT2ACYP3A4ALDH1A1CYP19A1
SCHEMBL29105124 0.85 HSP90AA1 (0.40) HSP90AA1KMT2ACYP3A4ALDH1A1CYP19A1
SCHEMBL9422845 0.84 HSP90AA1 (0.41) HSP90AA1KMT2ACYP3A4ALDH1A1CYP19A1
SCHEMBL9667126 0.84 HSP90AA1 (0.41) HSP90AA1KMT2ACYP3A4ALDH1A1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3762369-B1 A PROCESS FOR PREPARATION OF FUNGICIDALLY ACTIVE TRIAZOLE COMPOUNDS UPL LTD (IN) 2024-12-11 EP claimed
CN-112204016-B Process for preparing fungicidally active triazole compounds UPL有限公司 2024-06-21 CN claimed
CN-116655548-A Synthesis method of prothioconazole 河北八亿时空药业有限公司 2023-08-29 CN claimed
EP-4558488-A1 CRYSTALLINE FORMS OF 1,2,4-OXADIAZOLE FUNGICIDES Syngenta Crop Protection AG (CH) 2025-05-28 EP disclosed
CN-119677724-A Crystalline forms of 1,2, 4-oxadiazole fungicides 先正达农作物保护股份公司 2025-03-21 CN disclosed
EP-3762369-B1 A PROCESS FOR PREPARATION OF FUNGICIDALLY ACTIVE TRIAZOLE COMPOUNDS UPL LTD (IN) 2024-12-11 EP disclosed
CN-114501994-B Aqueous composition, method for preparing said composition and use thereof 世科姆奥克松股份公司 2024-10-29 CN disclosed
CN-112204016-B Process for preparing fungicidally active triazole compounds UPL有限公司 2024-06-21 CN disclosed
WO-2024018016-A1 CRYSTALLINE FORMS OF 1,2,4-OXADIAZOLE FUNGICIDES SYNGENTA CROP PROTECTION AG (CH) 2024-01-25 WO disclosed
CN-114085126-B Radioisotope carbon-14 marked benzyl compound, prothioconazole and preparation method and application thereof in metabolic experiment 张北北九食品检验技术有限公司 2023-09-29 CN disclosed
EP-4247796-A1 PROCESS FOR THE PREPARATION OF PROTHIOCONAZOLE AND INTERMEDIATES THEREOF ADAMA MAKHTESHIM LTD. (IL) 2023-09-27 EP disclosed
EP-4045488-A1 AN INDUSTRIAL SCALE PROCESS FOR THE PREPARATION OF PROTHIOCONAZOLE Hikal Limited (IN) 2022-08-24 EP disclosed
EP-4009787-A1 FUNGICIDE COMPOSITION SIPCAM OXON S.p.A. (IT) 2022-06-15 EP disclosed
CN-111093374-B STABILIZED PROSTABILIZER-CONTAINING FORMULATIONS WITH LOW 2- (1-CHLOROCYCLOPROPYL) -1- (2-CHLOROPHENYL) -3- (1H-1,2, 4-TRIAZOL-1-YL) PROPAN-2-OL CONTENT 拜耳股份公司 2022-06-10 CN disclosed
CN-111093374-B STABILIZED PROSTABILIZER-CONTAINING FORMULATIONS WITH LOW 2- (1-CHLOROCYCLOPROPYL) -1- (2-CHLOROPHENYL) -3- (1H-1,2, 4-TRIAZOL-1-YL) PROPAN-2-OL CONTENT 拜耳股份公司 2022-06-10 CN disclosed
CN-111093374-B STABILIZED PROSTABILIZER-CONTAINING FORMULATIONS WITH LOW 2- (1-CHLOROCYCLOPROPYL) -1- (2-CHLOROPHENYL) -3- (1H-1,2, 4-TRIAZOL-1-YL) PROPAN-2-OL CONTENT 拜耳股份公司 2022-06-10 CN disclosed
WO-2022107139-A1 PROCESS FOR THE PREPARATION OF PROTHIOCONAZOLE AND INTERMEDIATES THEREOF ADAMA MAKHTESHIM LTD. (IL) 2022-05-27 WO disclosed
CN-114501994-A Fungicidal composition 世科姆奥克松股份公司 2022-05-13 CN disclosed
WO-2022058522-A1 STABILIZATION OF THIOKETONES ON SURFACES BAYER AKTIENGESELLSCHAFT (DE) 2022-03-24 WO disclosed
CN-114085126-A Radioisotope carbon-14 labeled benzyl compound, prothioconazole, preparation method thereof and application thereof in metabolic experiment 张北北九食品检验技术有限公司 2022-02-25 CN disclosed