SCHEMBL29405503

SCHEMBL29405503

CC(C)(C)OC(=O)N1CCc2c(ccc(Br)c2F)C1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.55
NR1H2 P55055 1/20 0.54
ABHD6 Q9BV23 6/20 0.47
MAPK1 P28482 1/20 0.45
MKNK1 Q9BUB5 3/20 0.44
UCHL1 P09936 2/20 0.43
ADORA1 P30542 1/20 0.43
MAPT P10636 2/20 0.42
KDM4E B2RXH2 1/20 0.42
SCN9A Q15858 1/20 0.41
HDAC1 Q13547 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19642882 1.00 ESR2 (0.55) ESR2NR1H2ABHD6MAPK1MKNK1
SCHEMBL22993468 0.90 ESR2 (0.55) ESR2NR1H2ABHD6MAPK1MKNK1
SCHEMBL29391872 0.90 ESR2 (0.55) ESR2NR1H2ABHD6MAPK1MKNK1
SCHEMBL29697653 0.90 ESR2 (0.55) ESR2NR1H2ABHD6MAPK1MKNK1
SCHEMBL31159106 0.88 HDAC1 (0.46) ESR2NR1H2ABHD6MAPK1MKNK1
SCHEMBL19948765 0.85 ESR2 (0.55) ESR2NR1H2ABHD6MAPK1MKNK1
SCHEMBL4165540 0.85 NR1H2 (0.60) ESR2NR1H2ABHD6MAPK1UCHL1
SCHEMBL31067476 0.85 NR1H2 (0.60) ESR2NR1H2ABHD6MAPK1UCHL1
SCHEMBL29446113 0.85 ESR2 (0.55) ESR2NR1H2ABHD6MAPK1MKNK1
SCHEMBL15503058 0.84 ESR2 (0.52) ESR2NR1H2ABHD6MAPK1MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114206852-A Plasma kallikrein inhibitors 卡尔维斯塔制药有限公司 2022-03-18 CN disclosed