SCHEMBL2941003

SCHEMBL2941003

CC1(C)C(=O)N(c2ccc(SC(F)(F)F)cc2)C(=O)N1Cc1ccnc(Nc2ccc(C(=O)O)nc2)c1

nearest known ligand 0.77

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 19/20 0.77
PPARG P37231 1/20 0.41
PPARD Q03181 1/20 0.41
PPARA Q07869 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3734038 0.92 IGF1R (0.72) IGF1RPPARGPPARDPPARA
SCHEMBL4101203 0.90 IGF1R (0.78) IGF1R
SCHEMBL2935582 0.89 IGF1R (0.79) IGF1R
SCHEMBL4033708 0.88 IGF1R (0.78) IGF1R
SCHEMBL2939085 0.87 IGF1R (1.00) IGF1R
SCHEMBL2935176 0.87 IGF1R (0.75) IGF1R
SCHEMBL2941516 0.87 IGF1R (0.70) IGF1RPPARGPPARDPPARA
SCHEMBL13904188 0.86 IGF1R (0.80) IGF1R
SCHEMBL2939265 0.86 IGF1R (0.84) IGF1R
SCHEMBL4099471 0.86 IGF1R (0.81) IGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1599464-B1 NOVEL CYCLIC UREA DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL USE OF SAME AS KINASE INHIBITORS AVENTIS PHARMA SA (FR) 2010-09-22 EP claimed