SCHEMBL29439711

SCHEMBL29439711

COc1ncc(C(F)(F)F)cc1N

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2C19 P33261 1/20 0.54
MAPT P10636 2/20 0.49
CASP1 P29466 1/20 0.49
AURKA O14965 1/20 0.47
TTK P33981 1/20 0.47
AURKB Q96GD4 1/20 0.47
INCENP Q9NQS7 1/20 0.47
HPGD P15428 1/20 0.44
RAB9A P51151 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
KMT2A Q03164 2/20 0.41
PIK3CA P42336 1/20 0.40
METAP2 P50579 1/20 0.40
CFTR P13569 2/20 0.40
LMNA P02545 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18337425 1.00 CYP1A2 (0.54) CYP1A2CYP3A4CYP2C19MAPTCASP1
SCHEMBL84376 0.83 MAPT (0.50) CYP1A2CYP3A4CYP2C19MAPTCASP1
SCHEMBL15716504 0.82 CYP1A2 (0.45) CYP1A2CYP3A4CYP2C19HPGDKMT2A
SCHEMBL8427120 0.81 KMT2A (0.47) CYP1A2CYP3A4CYP2C19HPGDRAB9A
SCHEMBL10459325 0.79 CYP1A2 (0.48) CYP1A2CYP3A4CYP2C19MAPTAURKA
SCHEMBL38661825 0.79 CYP1A2 (0.44) CYP1A2CYP3A4CYP2C19HPGDRAB9A
SCHEMBL27906036 0.79 CYP1A2 (0.44) CYP1A2CYP3A4CYP2C19HPGDRAB9A
SCHEMBL27889651 0.78 CYP2C19 (0.45) CYP1A2CYP3A4CYP2C19MAPTHPGD
SCHEMBL7917526 0.78 CYP1A2 (0.43) CYP1A2CYP3A4CYP2C19HPGDRAB9A
SCHEMBL769495 0.78 CYP1A2 (0.61) CYP1A2CYP3A4CYP2C19HPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118908957-A Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-11-08 CN disclosed
CN-114222737-B Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-07-26 CN disclosed
EP-3976597-A1 SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE Janssen Pharmaceutica NV (BE) 2022-04-06 EP disclosed
CN-114222737-A Small molecule inhibitor of NF-kB induced kinase 詹森药业有限公司 2022-03-22 CN disclosed