SCHEMBL29444159

SCHEMBL29444159

C=CC(=O)N1CCC(Oc2cc3c(Nc4ccc(Cl)c(Cl)c4)c(C#N)cnc3cc2OC)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 12/20 1.00
EGFR P00533 16/20 0.88
SRC P12931 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22590126 1.00 ERBB2 (1.00) ERBB2EGFRSRC
SCHEMBL29444165 1.00 ERBB2 (1.00) ERBB2EGFRSRC
SCHEMBL29752032 0.94 EGFR (1.00) ERBB2EGFR
SCHEMBL22598672 0.94 EGFR (1.00) ERBB2EGFR
SCHEMBL22598775 0.93 ERBB2 (0.87) ERBB2EGFRSRC
SCHEMBL29752078 0.93 ERBB2 (0.87) ERBB2EGFRSRC
SCHEMBL22598674 0.92 EGFR (1.00) ERBB2EGFRSRC
SCHEMBL29751985 0.92 EGFR (1.00) ERBB2EGFRSRC
SCHEMBL22590135 0.92 ERBB2 (0.84) ERBB2EGFRSRC
SCHEMBL22598685 0.91 EGFR (1.00) ERBB2EGFRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118852118-A Compounds that inhibit tyrosine kinase activity and pharmaceutical compositions comprising the same 德州大学系统董事会 2024-10-29 CN disclosed
CN-114026083-B Heterocyclic inhibitors of tyrosine kinases 德州大学系统董事会 2024-07-09 CN disclosed
EP-3962908-A1 HETEROCYCLIC INHIBITORS OF TYROSINE KINASE Board of Regents, The University of Texas System (US) 2022-03-09 EP disclosed
CN-114026083-A Heterocyclic inhibitors of tyrosine kinases 德州大学系统董事会 2022-02-08 CN disclosed