SCHEMBL29447334

SCHEMBL29447334

Cc1ccccc1S(=O)(=O)Nc1c(CO[Si](C)(C)C(C)(C)C)cccc1CO[Si](C)(C)C(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
TP53 P04637 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
EDNRA P25101 2/20 0.44
EDNRB P24530 1/20 0.42
SLC40A1 Q9NP59 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MAPT P10636 1/20 0.41
BACE1 P56817 1/20 0.41
BRD4 O60885 1/20 0.40
PKM P14618 1/20 0.40
KDM4E B2RXH2 2/20 0.39
HPGD P15428 2/20 0.39
TAS2R8 Q9NYW2 1/20 0.39
POLB P06746 2/20 0.38
GFER P55789 1/20 0.38
PTPN2 P17706 3/20 0.38
PTPN1 P18031 3/20 0.38
PTPN5 P54829 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11220197 0.77 MAPT (0.52) ALDH1A1TP53TDP1EDNRAEDNRB
SCHEMBL5467148 0.72 BACE1 (0.39) ALDH1A1MAPTBACE1KDM4E
SCHEMBL7391015 0.72 BACE1 (0.44) ALDH1A1BACE1PKMKDM4EHPGD
SCHEMBL22498312 0.70 CA12 (0.43) ALDH1A1MAPTPKMPOLBHTT
SCHEMBL4680048 0.70 BACE1 (0.40) ALDH1A1BACE1KDM4EPOLB
SCHEMBL20558194 0.70 BACE1 (0.38) BACE1
SCHEMBL30703393 0.69 BACE1 (0.39) MAPTBACE1HPGD
SCHEMBL25897373 0.69 BACE1 (0.39) MAPTBACE1HPGD
SCHEMBL29387450 0.68 BACE1 (0.48) MAPTBACE1HPGD
SCHEMBL15389825 0.68 BACE1 (0.42) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3947344-A1 AMINOGUANIDINE HYDRAZONES AS RETROMER STABILIZERS USEFUL FOR TREATING NEUROLOGICAL DISEASES Ospedale San Raffaele Srl (IT) 2022-02-09 EP disclosed